SCHEMBL14201152

SCHEMBL14201152

CCCC(CCC)N(C(=O)C(C)C(C)(C)C)c1cccc(CC)c1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.36
SIGMAR1 Q99720 9/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPK1 P28482 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
TSHR P16473 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
EPHX1 P07099 1/20 0.34
BCL2 P10415 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14201150 0.91 PTGS2 (0.35) PTGS2SIGMAR1ALDH1A1SMN1; SMN2MAPK1
SCHEMBL14201127 0.86 TAS1R3 (0.43) ALDH1A1SMN1; SMN2TDP1TAS1R3TAS1R1
SCHEMBL14201120 0.85 MAPK1 (0.35) PTGS2SIGMAR1ALDH1A1SMN1; SMN2MAPK1
SCHEMBL14201110 0.85 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2TAS1R3TAS1R1
SCHEMBL14229313 0.84 PTGS2 (0.37) PTGS2SIGMAR1MAPK1L3MBTL1TSHR
SCHEMBL14201165 0.81 ALDH1A1 (0.36) PTGS2SIGMAR1ALDH1A1SMN1; SMN2MAPK1
SCHEMBL14229594 0.81 RIPK1 (0.43) SIGMAR1ALDH1A1SMN1; SMN2MAPK1L3MBTL1
SCHEMBL14200467 0.81 MAPK1 (0.37) PTGS2SIGMAR1ALDH1A1SMN1; SMN2MAPK1
SCHEMBL14229027 0.79 TP53 (0.42) PTGS2SIGMAR1MAPK1L3MBTL1TSHR
SCHEMBL14201177 0.79 RIPK1 (0.34) TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed