SCHEMBL142106

SCHEMBL142106

O=Cc1ccc(-c2ccc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c3c2)o1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.79
ERBB2 P04626 15/20 0.79
ABL1 P00519 4/20 0.79
INSR P06213 4/20 0.79
PDGFRB P09619 4/20 0.79
CDK2 P24941 4/20 0.79
PLK1 P53350 3/20 0.79
HDAC3 O15379 2/20 0.79
HDAC4 P56524 2/20 0.79
HDAC1 Q13547 2/20 0.79
HDAC7 Q8WUI4 2/20 0.79
HDAC2 Q92769 2/20 0.79
HDAC10 Q969S8 2/20 0.79
HDAC11 Q96DB2 2/20 0.79
HDAC8 Q9BY41 2/20 0.79
HDAC6 Q9UBN7 2/20 0.79
HDAC9 Q9UKV0 2/20 0.79
HDAC5 Q9UQL6 2/20 0.79
MEN1 O00255 1/20 0.71
PIK3C2B O00750 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29387336 1.00 EGFR (0.79) EGFRERBB2ABL1INSRPDGFRB
Hydrochloric Acid SCHEMBL2511570 0.99 EGFR (0.78) EGFRERBB2ABL1INSRPDGFRB
SCHEMBL1448581 0.94 EGFR (0.77) EGFRERBB2ABL1INSRPDGFRB
SCHEMBL12727551 0.93 EGFR (0.69) EGFRERBB2ABL1INSRPDGFRB
SCHEMBL15000311 0.92 EGFR (0.68) EGFRERBB2ABL1INSRPDGFRB
SCHEMBL3326173 0.92 EGFR (0.68) EGFRERBB2ABL1INSRPDGFRB
SCHEMBL3009979 0.91 EGFR (0.69) EGFRERBB2ABL1INSRPDGFRB
SCHEMBL142111 0.91 EGFR (0.68) EGFRERBB2ABL1INSRPDGFRB
SCHEMBL12719625 0.91 EGFR (0.66) EGFRERBB2ABL1INSRPDGFRB
SCHEMBL13966850 0.91 EGFR (0.68) EGFRERBB2ABL1INSRPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 256 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118184927-A Polymer material carrier, preparation method thereof, polymer material carrier supported palladium nanoparticle and application 河北科技大学 2024-06-14 CN claimed
US-20120295928-A1 METHODS FOR DETECTING AND REDUCING IMPURITIES OF LAPATINIB AND SALTS THEREOF F.I.S. FABBRICA ITALIANA SINTETICI S.P.A. (IT) 2012-11-22 US claimed
EP-2489661-A1 Impurity of lapatinib and salts thereof F.I.S. Fabbrica Italiana Sintetici S.p.A. (IT) 2012-08-22 EP claimed
EP-1454907-B1 Quninazoline and pyridopyrimidine derivatives GLAXO GROUP LTD (GB) 2008-12-17 EP claimed
US-20080058519-A1 QUINAZOLINE DITOSYLATE SALT COMPOUNDS LEO OSPREY LIMITED (GB) 2008-03-06 US claimed
US-7109333-B2 Heterocyclic compounds SMITHKLINE BEECHAM CORPORATION (US) 2006-09-19 US claimed
US-20050130996-A1 Heterocyclic compounds NOVARTIS AG (CH) 2005-06-16 US claimed
EP-1454907-A1 Quninazoline and pyridopyrmidine derivatives Glaxo Group Limited (GB) 2004-09-08 EP claimed
US-12594275-B2 Immunophilin binding agents and uses thereof THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2026-04-07 US disclosed
US-12558356-B2 Immunophilin binding agents and uses thereof THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2026-02-24 US disclosed
US-20250108052-A1 IMMUNOPHILIN BINDING AGENTS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2025-04-03 US disclosed
CN-118184927-A Polymer material carrier, preparation method thereof, polymer material carrier supported palladium nanoparticle and application 河北科技大学 2024-06-14 CN disclosed
US-20230063768-A1 IMMUNOPHILIN BINDING AGENTS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2023-03-02 US disclosed
US-20230063768-A1 IMMUNOPHILIN BINDING AGENTS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2023-03-02 US disclosed
WO-2002056912-A2 PHARMACEUTICAL COMBINATION FOR THE TREATMENT OF CANCER CONTAINING A 4-QUINAZOLINEAMINE AND ANOTHER ANTI-NEOPLASTIC AGENT GLAXO GROUP LIMITED (GB) 2002-07-25 WO disclosed
EP-1192151-A1 ANILINOQUINAZOLINES AS PROTEIN TYROSINE KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2002-04-03 EP disclosed
WO-2002002552-A1 QUINAZOLINE DITOSYLATE SALT COMPOUNDS GLAXO GROUP LIMITED (GB) 2002-01-10 WO disclosed
WO-2001004111-A1 ANILINOQUINAZOLINES AS PROTEIN TYROSINE KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2001-01-18 WO disclosed
EP-1047694-A1 BICYCLIC HETEROAROMATIC COMPOUNDS AS PROTEIN TYROSINE KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2000-11-02 EP disclosed
WO-1999035146-A1 BICYCLIC HETEROAROMATIC COMPOUNDS AS PROTEIN TYROSINE KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 1999-07-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120295928-A1 METHODS FOR DETECTING AND REDUCING IMPURITIES OF LAPATINIB AND SALTS THEREOF SRMS, ABL1, ERBB2 EGFR 5/4885ERBB2 3/4885ABL1 2/4885
US-20080058519-A1 QUINAZOLINE DITOSYLATE SALT COMPOUNDS ERBB4, ABL1, ERBB2 EGFR 64/4885ERBB2 3/4885ABL1 2/4885
US-20230063768-A1 IMMUNOPHILIN BINDING AGENTS AND USES THEREOF PMP22, MAG, FABP7 EGFR 3726/4885ERBB2 3924/4885ABL1 4111/4885
US-12594275-B2 Immunophilin binding agents and uses thereof CCR1, CCRL2, CCR3 EGFR 2717/4885ERBB2 1975/4885ABL1 4373/4885
US-20050130996-A1 Heterocyclic compounds CCNH, SDHA, CYP1A2 EGFR 3748/4885ERBB2 3150/4885ABL1 1065/4885
US-20250108052-A1 IMMUNOPHILIN BINDING AGENTS AND USES THEREOF SERPINA6, SELPLG, FABP7 EGFR 3638/4885ERBB2 3961/4885ABL1 3639/4885
US-12558356-B2 Immunophilin binding agents and uses thereof CCRL2, CFB, CCR3 EGFR 1974/4885ERBB2 1701/4885ABL1 3756/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.