SCHEMBL1421794

SCHEMBL1421794

COc1cc(N(CCc2ccc(C(F)(F)F)nc2)C(=O)[C@](O)(c2ccc(F)cc2)[C@](O)(C(=O)N(CCc2ccc(C(F)(F)F)nc2)c2ccc(C)c(OC)c2)c2ccc(F)cc2)ccc1C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTC4S Q16873 1/20 0.35
GPBAR1 Q8TDU6 5/20 0.35
QPCT Q16769 4/20 0.35
PPARD Q03181 1/20 0.34
CSF1R P07333 2/20 0.34
NTRK1 P04629 1/20 0.34
NTRK2 Q16620 1/20 0.34
TRPA1 O75762 1/20 0.34
POLQ O75417 2/20 0.33
FFAR1 O14842 1/20 0.33
FFAR2 O15552 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
RORC P51449 1/20 0.33
MEN1 O00255 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL265374 0.84 CSF1R (0.38) LTC4SGPBAR1QPCTPPARDCSF1R
SCHEMBL265373 0.84 CSF1R (0.38) LTC4SGPBAR1QPCTPPARDCSF1R
SCHEMBL264165 0.78 GPBAR1 (0.37) GPBAR1PPARDCSF1R
SCHEMBL264166 0.78 GPBAR1 (0.37) GPBAR1PPARDCSF1R
SCHEMBL1422138 0.78 ALDH1A1 (0.33) GPBAR1PPARDMEN1CYP3A4CYP2D6
SCHEMBL1422511 0.76 TRPM8 (0.35) PPARDMEN1KMT2A
SCHEMBL1422515 0.76 TRPM8 (0.34) PPARDMEN1KMT2A
SCHEMBL1422609 0.76 GPBAR1 (0.34) LTC4SGPBAR1PPARDPOLQMEN1
SCHEMBL1422607 0.76 GPBAR1 (0.34) LTC4SGPBAR1PPARDPOLQMEN1
SCHEMBL265595 0.75 P2RX7 (0.39) PPARDTRPA1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2297102-A1 HETEROAROMATIC MONOAMIDES AS OREXININ RECEPTOR ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2011-03-23 EP disclosed