SCHEMBL14219656

SCHEMBL14219656

Cc1cnc(Nc2c(C(=O)NOC(C)(C)C)cc(Cl)c(F)c2F)c(C)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.41
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
LCK P06239 2/20 0.33
DHODH Q02127 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SCN9A Q15858 2/20 0.32
EGFR P00533 2/20 0.30
MAP2K1 Q02750 2/20 0.30
HTT P42858 1/20 0.30
SMC2 O95347 1/20 0.30
CSNK2A2 P19784 1/20 0.30
MAP2K2 P36507 1/20 0.30
SMC1A Q14683 1/20 0.30
AAK1 Q2M2I8 1/20 0.30
Q6ZSR9 Q6ZSR9 1/20 0.30
BMP2K Q9NSY1 1/20 0.30
IRAK4 Q9NWZ3 1/20 0.30
MEN1 O00255 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14220128 0.90 PTGS2 (0.37) PTGS2CNR1CNR2DHODHNPC1
SCHEMBL14219642 0.89 TDP1 (0.39) PTGS2LCKDHODHNPC1RAB9A
SCHEMBL14219717 0.87 PTGS2 (0.38) PTGS2CNR1CNR2SCN9AEGFR
SCHEMBL14219715 0.83 PTGS2 (0.41) PTGS2CNR1CNR2DHODHRAB9A
SCHEMBL14220130 0.83 ALDH1A1 (0.37) LCKDHODHNPC1RAB9AEGFR
SCHEMBL14219683 0.82 LMNA (0.42) LCKDHODHNPC1RAB9AMAP2K1
SCHEMBL14220117 0.81 MEN1 (0.51) SCN9AEGFRMAP2K1SMC2CSNK2A2
SCHEMBL14220114 0.81 PTGS2 (0.34) PTGS2DHODHEGFRMAP2K1IRAK4
SCHEMBL14223052 0.81 MAP2K1 (0.45) EGFRMAP2K1SMC2CSNK2A2MAP2K2
SCHEMBL14219843 0.81 MAP2K1 (0.45) EGFRMAP2K1SMC2CSNK2A2MAP2K2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1908751-A1 N-hydroxy benzamides with antitumour activity EOS S.p.A. (IT) 2008-04-09 EP disclosed