SCHEMBL14223271

SCHEMBL14223271

Nc1ccc(Cc2ccncc2I)c(F)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRA2B P18089 1/20 0.49
LOXL2 Q9Y4K0 1/20 0.41
AOC1 P19801 4/20 0.35
AOC3 Q16853 4/20 0.35
MAPT P10636 3/20 0.33
GAA P10253 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
MPO P05164 1/20 0.32
DPP4 P27487 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
PRKCZ Q05513 1/20 0.31
CYP17A1 P05093 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP19A1 P11511 1/20 0.30
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25577644 0.82 ADRA2B (0.49) ADRA2BLOXL2AOC1AOC3MAPT
SCHEMBL26037690 0.78 ADRA2B (0.50) ADRA2BMAPTGAATSHRMAPK1
SCHEMBL31175766 0.78 ADRA2B (0.50) ADRA2BMAPTGAATSHRMAPK1
SCHEMBL7215312 0.74 ADRA2B (0.47) ADRA2BLOXL2MAPTGAATSHR
SCHEMBL4731181 0.70 ROCK2 (0.36) ADRA2BCYP3A4
SCHEMBL2882589 0.69 ADRA2B (0.45) ADRA2BMPO
SCHEMBL26037444 0.68 GAA (0.44) ADRA2BMAPTGAATSHRMAPK1
SCHEMBL31175764 0.68 CYP3A4 (0.52) ADRA2BLOXL2MAPTGAATSHR
SCHEMBL10718351 0.68 CYP3A4 (0.52) ADRA2BLOXL2MAPTGAATSHR
SCHEMBL25318193 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008046216-A1 KINASE INHIBITORS AND USES THEREOF METHYLGENE, INC. (CA) 2008-04-24 WO disclosed