SCHEMBL14229095

SCHEMBL14229095

CCCCN(CCCC)C(=O)c1ccc(OC)cc1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.57
ERBB2 P04626 1/20 0.57
HPGD P15428 3/20 0.55
GAA P10253 1/20 0.55
LPAR1 Q92633 3/20 0.54
LPAR5 Q9H1C0 2/20 0.54
HDAC1 Q13547 2/20 0.51
HDAC3 O15379 1/20 0.51
HDAC2 Q92769 1/20 0.51
TSHR P16473 2/20 0.50
OPRM1 P35372 1/20 0.50
OPRD1 P41143 1/20 0.50
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
DRD2 P14416 1/20 0.48
LMNA P02545 1/20 0.48
MLYCD O95822 1/20 0.47
KDM4E B2RXH2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14229444 0.97 EGFR (0.55) EGFRERBB2HPGDGAALPAR1
SCHEMBL10144056 0.94 HPGD (0.64) EGFRERBB2HPGDGAALPAR1
SCHEMBL14200268 0.90 EGFR (0.49) EGFRERBB2HPGDGAALPAR1
SCHEMBL6674114 0.88 EGFR (0.70) EGFRERBB2HPGDGAAHDAC1
SCHEMBL27709184 0.86 BMP1 (0.52) HPGDGAALPAR1LPAR5HDAC1
SCHEMBL11213030 0.85 OPRM1 (0.56) HPGDGAALPAR1TSHROPRM1
SCHEMBL9888801 0.85 DRD2 (0.50) HPGDLPAR1LPAR5HDAC1OPRM1
SCHEMBL11757402 0.85 OPRM1 (0.56) HPGDGAALPAR1TSHROPRM1
SCHEMBL19997006 0.85 DRD2 (0.61) HPGDHDAC1HDAC3HDAC2CES2
SCHEMBL6023472 0.83 CES2 (0.52) HPGDLPAR1LPAR5HDAC1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106278775-A The preparation method of a kind of arylamides and purification method thereof 温州大学 2017-01-04 CN disclosed
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed