SCHEMBL14229592

SCHEMBL14229592

CCCC(C)N(C(=O)C(C)CC)c1cccc(CC)c1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.36
SIGMAR1 Q99720 9/20 0.36
TSHR P16473 2/20 0.34
MAPK1 P28482 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
BCL2 P10415 1/20 0.34
HSD17B10 Q99714 1/20 0.34
KAT6A Q92794 1/20 0.34
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14229559 0.91 MAPK1 (0.36) PTGS2SIGMAR1MAPK1L3MBTL1
SCHEMBL14229313 0.91 PTGS2 (0.37) PTGS2SIGMAR1TSHRMAPK1L3MBTL1
SCHEMBL14229004 0.85 TAS1R3 (0.44) TSHRTDP1HSD17B10
SCHEMBL14201150 0.85 PTGS2 (0.35) PTGS2SIGMAR1TSHRMAPK1L3MBTL1
SCHEMBL14229475 0.84 ALDH1A1 (0.39)
SCHEMBL14229349 0.83 TP53 (0.40) PTGS2SIGMAR1TSHRMAPK1L3MBTL1
SCHEMBL14230178 0.80 RIPK1 (0.41) PTGS2SIGMAR1
SCHEMBL14200447 0.80 MAPK1 (0.36) PTGS2SIGMAR1TSHRMAPK1L3MBTL1
SCHEMBL14201516 0.80 EPHX1 (0.36) PTGS2SIGMAR1TSHRMAPK1L3MBTL1
SCHEMBL14229086 0.78 GAA (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed