SCHEMBL14229686

SCHEMBL14229686

CCCCN(CCOC)S(=O)(=O)CC(C)C

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.35
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
PKM P14618 1/20 0.33
CYP2C19 P33261 1/20 0.33
MMP3 P08254 2/20 0.31
PER2 O15055 1/20 0.31
CRY1 Q16526 1/20 0.31
CRY2 Q49AN0 1/20 0.31
MAPK1 P28482 1/20 0.31
TP53 P04637 1/20 0.30
MMP1 P03956 1/20 0.30
MMP2 P08253 1/20 0.30
MMP8 P22894 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19766998 0.89 PIK3CD (0.42) PIK3CDPER2CRY1CRY2
SCHEMBL14229345 0.88 TP53 (0.36) MMP3TP53MMP1MMP2MMP8
SCHEMBL14229451 0.84 CA1 (0.43) TP53
SCHEMBL14230123 0.84 PIK3CD (0.37) PIK3CDCYP1A2CYP3A4CYP2C9PKM
SCHEMBL25456874 0.83 PIK3CD (0.37) PIK3CD
SCHEMBL14229149 0.81 BMP1 (0.41) CYP1A2CYP3A4CYP2C9PKMCYP2C19
SCHEMBL14229525 0.79 CNR2 (0.38) CYP1A2CYP3A4CYP2C9PKMCYP2C19
SCHEMBL14229124 0.79 MMP3 (0.36) MMP3TP53
SCHEMBL14200421 0.79 PIK3CD (0.34) PIK3CD
SCHEMBL14229340 0.78 CNR2 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed