SCHEMBL14249161

SCHEMBL14249161

OCC1(O)CCN(c2nc(-c3ccc(N4CCOCC4)nc3)c3nc[nH]c3n2)CC1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 12/20 0.42
PIK3R1 P27986 10/20 0.42
CNR2 P34972 4/20 0.39
KDM5B Q9UGL1 1/20 0.38
PIK3CD O00329 1/20 0.38
PIK3CB P42338 1/20 0.38
TDO2 P48775 1/20 0.38
ATR Q13535 1/20 0.38
ATRIP Q8WXE1 1/20 0.38
MTOR P42345 1/20 0.38
ADK P55263 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14249567 0.91 PIK3CA (0.46) PIK3CAPIK3R1PIK3CDPIK3CBMTOR
SCHEMBL14249549 0.82 MAP3K11 (0.34) PIK3CAPIK3R1PIK3CDPIK3CBATR
Hydrochloric Acid SCHEMBL14249557 0.81 PIK3CA (0.35) PIK3CAPIK3R1PIK3CDPIK3CBATR
SCHEMBL14316031 0.77 CNR2 (0.50) CNR2KDM5BTDO2ATRATRIP
SCHEMBL8079836 0.77 PIK3CA (0.59) PIK3CAPIK3R1PIK3CDPIK3CBATR
SCHEMBL8062292 0.77 PIK3CA (0.58) PIK3CAPIK3R1PIK3CDPIK3CBMTOR
SCHEMBL14249658 0.75 FLT3 (0.49) PIK3CAPIK3R1ATRMTOR
SCHEMBL12537215 0.74 ATR (0.49) PIK3CAPIK3R1ATRATRIPMTOR
SCHEMBL1568626 0.70 PIK3CA (0.65) PIK3CAMTOR
SCHEMBL27784940 0.70 ADORA3 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012172043-A1 PURINE DERIVATIVES AND THEIR USE AS PHARMACEUTICALS FOR PREVENTION OR TREATMENT OF BACTERIAL INFECTIONS LABORATOIRE BIODIM (FR) 2012-12-20 WO disclosed
WO-2012172043-A1 PURINE DERIVATIVES AND THEIR USE AS PHARMACEUTICALS FOR PREVENTION OR TREATMENT OF BACTERIAL INFECTIONS LABORATOIRE BIODIM (FR) 2012-12-20 WO disclosed