SCHEMBL14276271

SCHEMBL14276271

CCOC(=O)c1cc2cccc(Oc3ccnc(Cl)n3)c2n1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.39
NOD2 Q9HC29 5/20 0.38
NOD1 Q9Y239 5/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
MAPT P10636 4/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
GPR119 Q8TDV5 1/20 0.38
KDM4E B2RXH2 3/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP1A2 P05177 1/20 0.36
GABRA2 P47869 1/20 0.36
GABRB2 P47870 1/20 0.36
MAPK1 P28482 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
ALDH1A1 P00352 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14276270 0.87 KDR (0.39) MAPK14NOD2NOD1SMN1; SMN2MAPT
SCHEMBL4049497 0.84 PPARG (0.41) NOD2NOD1SMN1; SMN2MAPTNPC1
SCHEMBL14276263 0.80 P2RX3 (0.39) SMN1; SMN2MAPTNPC1RAB9AKDM4E
SCHEMBL14376280 0.78 PPARG (0.48) NOD2NOD1CYP1A2
SCHEMBL7884857 0.78 KMT2A (0.47) NOD2NOD1SMN1; SMN2MAPTKDM4E
SCHEMBL14276261 0.77 BRAF (0.45)
SCHEMBL3052830 0.77 NOD2 (0.46) NOD2NOD1SMN1; SMN2MAPTNPC1
SCHEMBL14276284 0.77 SMN1; SMN2 (0.34) NOD2NOD1SMN1; SMN2MAPTNPC1
SCHEMBL30220535 0.77 JMJD6 (0.41) NOD2NOD1SMN1; SMN2MAPTNPC1
SCHEMBL13690239 0.77 TP53 (0.41) NOD2NOD1SMN1; SMN2MAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7335657-B2 Cytokine inhibitors BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2008-02-26 US disclosed
US-7335657-B2 Cytokine inhibitors BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2008-02-26 US disclosed