SCHEMBL142843

SCHEMBL142843

CSc1nc(=O)cc(CCl)[nH]1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.41
POLB P06746 1/20 0.39
HTT P42858 2/20 0.39
KDM4E B2RXH2 2/20 0.37
MAPT P10636 2/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 2/20 0.35
GAA P10253 1/20 0.34
KDM6B O15054 1/20 0.33
KDM4A O75164 1/20 0.33
KDM4D Q6B0I6 1/20 0.33
HIF1AN Q9NWT6 1/20 0.33
KDM2A Q9Y2K7 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23160932 0.84 HTT (0.47) PKMPOLBHTTKDM4EMAPT
SCHEMBL9878843 0.81 ADORA1 (0.44) PKMPOLBHTTKDM4EMAPT
SCHEMBL798506 0.79 PKM (0.58) PKMPOLBHTTKDM4EMAPT
SCHEMBL9878574 0.76 POLB (0.61) POLBHTTKDM4ESMN1; SMN2HPGD
SCHEMBL29232331 0.76 SMN1; SMN2 (0.52) HTTKDM4EMAPTSMN1; SMN2HPGD
SCHEMBL9697629 0.73 MAPT (0.60) PKMPOLBHTTKDM4EMAPT
SCHEMBL5124123 0.72 PKM (0.41) PKMPOLBHTTKDM4EMAPT
SCHEMBL117000 0.72 PKM (0.41) PKMPOLBHTTKDM4EMAPT
SCHEMBL17594977 0.72 PKM (0.41) PKMPOLBHTTKDM4EMAPT
SCHEMBL10852387 0.71 HCAR2 (0.37) PKMHTTKDM4ESMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3759082-B1 PROCESS FOR THE SYNTHESIS OF 6-CHLOROMETHYLURACIL PROCOS SPA (IT) 2022-04-20 EP claimed
US-11028057-B2 Process for the synthesis of 6-chloromethyluracil PROCOS S.P.A. (IT) 2021-06-08 US claimed
EP-3759082-A1 PROCESS FOR THE SYNTHESIS OF 6-CHLOROMETHYLURACIL Procos S.p.A. (IT) 2021-01-06 EP claimed
US-20200407330-A1 PROCESS FOR THE SYNTHESIS OF 6-CHLOROMETHYLURACIL PROCOS S.P.A. (IT) 2020-12-31 US claimed
EP-3759082-B1 PROCESS FOR THE SYNTHESIS OF 6-CHLOROMETHYLURACIL PROCOS SPA (IT) 2022-04-20 EP disclosed
EP-3759082-B1 PROCESS FOR THE SYNTHESIS OF 6-CHLOROMETHYLURACIL PROCOS SPA (IT) 2022-04-20 EP disclosed
US-11028057-B2 Process for the synthesis of 6-chloromethyluracil PROCOS S.P.A. (IT) 2021-06-08 US disclosed
US-11028057-B2 Process for the synthesis of 6-chloromethyluracil PROCOS S.P.A. (IT) 2021-06-08 US disclosed
EP-3759082-A1 PROCESS FOR THE SYNTHESIS OF 6-CHLOROMETHYLURACIL Procos S.p.A. (IT) 2021-01-06 EP disclosed
US-20200407330-A1 PROCESS FOR THE SYNTHESIS OF 6-CHLOROMETHYLURACIL PROCOS S.P.A. (IT) 2020-12-31 US disclosed
US-20200407330-A1 PROCESS FOR THE SYNTHESIS OF 6-CHLOROMETHYLURACIL PROCOS S.P.A. (IT) 2020-12-31 US disclosed
US-20120058984-A1 PYRIMIDINE DERIVATIVES USED AS ITK INHIBITORS GLAXO GROUP LIMITED (GB) 2012-03-08 US disclosed
EP-2408769-A1 PYRIMIDINE DERIVATIVES USED AS ITK INHIBITORS Glaxo Group Limited (GB) 2012-01-25 EP disclosed
WO-2010106016-A1 PYRIMIDINE DERIVATIVES USED AS ITK INHIBITORS GLAXO GROUP LIMITED (GB) 2010-09-23 WO disclosed
US-4604466-A INTERMEDIATES FOR BRONCHODILATORS RIKER LABORATORIES, INC. (US) 1986-08-05 US disclosed
US-4478835-A BRONCHODILATORS RIKER LABORATORIES, INC. (US) 1984-10-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120058984-A1 PYRIMIDINE DERIVATIVES USED AS ITK INHIBITORS DTYMK, ITK, DCK PKM 538/4885POLB 397/4885HTT 4389/4885
US-11028057-B2 Process for the synthesis of 6-chloromethyluracil DHPS, TPMT, MPST PKM 1409/4885POLB 209/4885HTT 1906/4885
US-20200407330-A1 PROCESS FOR THE SYNTHESIS OF 6-CHLOROMETHYLURACIL DHPS, TPMT, MPST PKM 1409/4885POLB 209/4885HTT 1906/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.