SCHEMBL14600752

SCHEMBL14600752

NC(=O)c1nc(-c2conc2-c2cccc(F)c2F)c[nH]1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.36
RAB9A P51151 4/20 0.36
CCNE2 O96020 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
SLC9A1 P19634 3/20 0.33
PARP1 P09874 1/20 0.33
LRRK2 Q5S007 1/20 0.32
GRK6 P43250 1/20 0.32
JAK2 O60674 1/20 0.32
CDC7 O00311 1/20 0.32
DBF4 Q9UBU7 1/20 0.32
PIM1 P11309 1/20 0.31
PIM3 Q86V86 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
DHODH Q02127 1/20 0.31
MAOA P21397 1/20 0.30
BLVRB P30043 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14600754 0.83 HPGD (0.42) NPC1RAB9ACCNE2CCNE1CDK2
SCHEMBL14600758 0.79 GSK3B (0.41) NPC1RAB9A
SCHEMBL14286128 0.77 CCNC (0.41) NPC1RAB9ACCNE2CCNE1CDK2
SCHEMBL14600757 0.76 ALDH1A1 (0.44) NPC1RAB9A
SCHEMBL14600755 0.66 BCAT1 (0.41) NPC1RAB9ACCNE2CCNE1CDK2
SCHEMBL7438138 0.66 HPGDS (0.54) CDK2SLC9A1PARP1CDC7PIM1
SCHEMBL14600775 0.65 BCAT1 (0.39) RAB9ACCNE2CCNE1CDK2SLC9A1
SCHEMBL4243696 0.63 MAP2K3 (0.47) NPC1RAB9APARP1DHODH
SCHEMBL14564382 0.61 DHODH (0.50) CDK2PARP1CDC7PIM1PIM3
SCHEMBL15059858 0.61 NPC1 (0.55) NPC1RAB9ASLC9A1PARP1JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7169800-B2 Imidazole compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-01-30 US disclosed
US-7169800-B2 Imidazole compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-01-30 US disclosed