SCHEMBL14286159

SCHEMBL14286159

O=C(NCC1CCCC1)c1cc(-n2nnnc2-c2c(F)cccc2Cl)c[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
CHRM1 P11229 4/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
PTGES O14684 1/20 0.39
CHRM3 P20309 1/20 0.38
P2RX7 Q99572 2/20 0.38
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
MDM2 Q00987 1/20 0.37
MAPK14 Q16539 1/20 0.36
CRHR1 P34998 1/20 0.35
RIPK1 Q13546 1/20 0.35
IL1B P01584 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10067970 0.83 PTGES (0.39) ALDH1A1LMNACHRM1NPC1RAB9A
SCHEMBL14286151 0.80 ADORA2A (0.39) CHRM1NPC1RAB9AADORA2AADORA1
SCHEMBL14600765 0.71 ADORA2A (0.41) NPC1RAB9APTGESADORA2AADORA1
SCHEMBL14286139 0.67 ROCK2 (0.40) CHRM1ADORA2AADORA1MAPK14MEN1
SCHEMBL14286160 0.66 CHRM1 (0.42) CHRM1NPC1RAB9ACHRM3ADORA2A
SCHEMBL14286138 0.64 GSK3B (0.45) CHRM1CHRM3ADORA2AADORA1MEN1
SCHEMBL14286135 0.64 ROCK2 (0.41) CHRM1ADORA2AADORA1MAPK14MEN1
SCHEMBL15551944 0.64 CHRM1 (0.42) LMNACHRM1CHRM3P2RX7CNR1
SCHEMBL14286161 0.63 ALDH1A1 (0.36) ALDH1A1LMNAPTGESMAPK14MEN1
SCHEMBL14286176 0.63 HPGD (0.52) ALDH1A1LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7314885-B2 Pyrrole compounds useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-01-01 US disclosed
US-7314885-B2 Pyrrole compounds useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-01-01 US disclosed