SCHEMBL14286161

SCHEMBL14286161

O=C(Nc1ncc[nH]1)c1cc(-n2nnnc2-c2cccc(F)c2F)c[nH]1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 1/20 0.36
MAPK7 Q13164 8/20 0.36
MAPK14 Q16539 5/20 0.36
KCNN4 O15554 6/20 0.34
CYP3A4 P08684 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
PTGES O14684 1/20 0.32
YTHDC1 Q96MU7 1/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10067972 0.82 KCNN4 (0.34) ALDH1A1KMT2ALMNAKCNN4PTGES
SCHEMBL5042176 0.78 ALDH1A1 (0.39) ALDH1A1KMT2ALMNAKCNN4CYP3A4
SCHEMBL14286146 0.73 ADRA2A (0.37) MAPK7MAPK14PTGES
SCHEMBL14286152 0.73 MAPK7 (0.37) MAPK7MAPK14PTGESYTHDC1
SCHEMBL14310378 0.70 PTGES (0.37) ALDH1A1KMT2ALMNAMAPK7CYP3A4
SCHEMBL14286141 0.65 NPC1 (0.47) KMT2ALMNAMEN1POLB
SCHEMBL14600769 0.65 CCNE2 (0.34) PTGES
SCHEMBL14600771 0.64 ADRA2A (0.37) ALDH1A1KMT2ALMNAPTGES
SCHEMBL14286159 0.63 ALDH1A1 (0.41) ALDH1A1KMT2ALMNAMAPK14PTGES
SCHEMBL14278719 0.63 OPRD1 (0.37) ALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7314885-B2 Pyrrole compounds useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-01-01 US disclosed