SCHEMBL14288685

SCHEMBL14288685

Cc1cc(C)c(N2CCN(c3ccccc3)CC2)c(C)c1NS(=O)(=O)c1ccc(C(C)(C)C)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 4/20 0.45
MAPT P10636 2/20 0.43
GLA P06280 1/20 0.43
ATM Q13315 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
UQCRB P14927 2/20 0.43
HSD17B2 P37059 4/20 0.42
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
FFAR4 Q5NUL3 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
NPC1 O15118 1/20 0.41
MAPK1 P28482 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL533091 0.88 BRPF1 (0.52) MAPTUQCRBHSD17B2MEN1LMNA
SCHEMBL532836 0.83 HSD17B2 (0.42) MAPTTDP1UQCRBHSD17B2MEN1
SCHEMBL14288683 0.82 RAD52 (0.53) MAPTTDP1MEN1LMNAHTT
SCHEMBL532776 0.80 FFAR4 (0.54) MAPTTDP1MEN1LMNAKMT2A
SCHEMBL534077 0.78 TSHR (0.47) HSD11B1MAPTMEN1LMNAKMT2A
SCHEMBL14288684 0.77 ACLY (0.53)
SCHEMBL533017 0.75 FFAR4 (0.55) MAPTTDP1MEN1LMNAKMT2A
SCHEMBL10092382 0.74 FFAR4 (0.53) MAPTATMLMNAKMT2AFFAR4
SCHEMBL533666 0.73 FFAR4 (0.56) MAPTMEN1LMNAHTTKMT2A
SCHEMBL533055 0.73 ALDH1A1 (0.45) MAPTTDP1MEN1KMT2AFFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed