SCHEMBL143083

SCHEMBL143083

O=C(C=Cc1ccccc1)NC(=O)c1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.66
NPC1 O15118 2/20 0.66
RAB9A P51151 2/20 0.66
TDP1 Q9NUW8 1/20 0.66
HDAC1 Q13547 7/20 0.63
HDAC3 O15379 6/20 0.63
HDAC4 P56524 5/20 0.63
HDAC2 Q92769 5/20 0.63
HDAC8 Q9BY41 5/20 0.63
HDAC6 Q9UBN7 5/20 0.63
HTT P42858 1/20 0.62
KMT2A Q03164 1/20 0.59
MAOB P27338 2/20 0.58
RECQL P46063 2/20 0.58
PLIN1 O60240 1/20 0.58
LMNA P02545 1/20 0.58
BCHE P06276 1/20 0.58
TNFRSF1A P19438 1/20 0.58
ACHE P22303 1/20 0.58
PLIN5 Q00G26 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7666658 1.00 MAPT (0.66) MAPTNPC1RAB9ATDP1HDAC1
SCHEMBL5425525 0.89 HDAC3 (0.54) MAPTNPC1RAB9ATDP1HDAC1
SCHEMBL8562018 0.89 NPC1 (0.57) MAPTNPC1RAB9ATDP1HDAC1
SCHEMBL5425520 0.89 HDAC3 (0.54) MAPTNPC1RAB9ATDP1HDAC1
SCHEMBL29060766 0.86 HDAC2 (0.76) MAPTNPC1RAB9ATDP1HDAC1
SCHEMBL4029206 0.86 HDAC2 (0.76) MAPTNPC1RAB9ATDP1HDAC1
SCHEMBL8559227 0.85 ALDH1A1 (0.78) MAPTNPC1RAB9ATDP1HDAC1
SCHEMBL9177259 0.85 EGFR (0.55) MAPTNPC1RAB9ATDP1HDAC1
SCHEMBL9177257 0.85 EGFR (0.55) MAPTNPC1RAB9ATDP1HDAC1
SCHEMBL28440928 0.84 HDAC2 (0.73) MAPTNPC1RAB9ATDP1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116606247-A Imide compound and preparation method and application thereof 温州医科大学 2023-08-18 CN disclosed
CN-107162928-B Halogenated analogs of anti-fibrotic agents 塞尔塔医疗有限公司 2022-03-11 CN disclosed
EP-3045170-B1 HALOGENATED ANALOGUES OF ANTI-FIBROTIC AGENTS FIBROTECH THERAPEUTICS PTY LTD (AU) 2018-07-04 EP disclosed
CN-107162928-A The halogenated analogues of antifibrotic agents 法博太科制药有限公司 2017-09-15 CN disclosed
EP-3045170-A1 HALOGENATED ANALOGUES OF ANTI-FIBROTIC AGENTS Fibrotech Therapeutics PTY LTD (AU) 2016-07-20 EP disclosed
EP-2220028-B1 HALOGENATED ANALOGUES OF ANTI-FIBROTIC AGENTS FIBROTECH THERAPEUTICS PTY LTD (AU) 2016-03-09 EP disclosed
US-8624056-B2 Halogenated analogues of anti-fibrotic agents FIBROTECH THERAPEUTICS PTY LTD 2014-01-07 US disclosed
US-20120059188-A9 HALOGENATED ANALOGUES OF ANTI-FIBROTIC AGENTS THE UNIVERSITY OF MELBOURNE (AU) 2012-03-08 US disclosed
US-20110021815-A1 HALOGENATED ANALOGUES OF ANTI-FIBROTIC AGENTS FIBROTECH THERAPEUTICS PTY LTD (AU) 2011-01-27 US disclosed
WO-2010144959-A1 ANALOGUES OF ANTI-FIBROTIC AGENTS FIBROTECH THERAPEUTICS PTY LTD (AU) 2010-12-23 WO disclosed
EP-2220028-A1 HALOGENATED ANALOGUES OF ANTI-FIBROTIC AGENTS Fibrotech Therapeutics PTY LTD (AU) 2010-08-25 EP disclosed
WO-2009079692-A1 HALOGENATED ANALOGUES OF ANTI-FIBROTIC AGENTS FIBROTECH THERAPEUTICS PTY LTD (AU) 2009-07-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120059188-A9 HALOGENATED ANALOGUES OF ANTI-FIBROTIC AGENTS MMP1, FIBP, HDGF MAPT 4850/4885NPC1 1501/4885RAB9A 1799/4885
US-20110021815-A1 HALOGENATED ANALOGUES OF ANTI-FIBROTIC AGENTS MMP1, FIBP, HDGF MAPT 4850/4885NPC1 1501/4885RAB9A 1799/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.