SCHEMBL14334255

SCHEMBL14334255

NC(=O)c1cccnc1O[C@@H]1CCCNC1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 2/20 0.58
CHEK1 O14757 1/20 0.54
KCNH2 Q12809 1/20 0.54
CHRNB2 P17787 1/20 0.49
CHRNA4 P43681 1/20 0.49
ROCK2 O75116 14/20 0.48
MKNK1 Q9BUB5 1/20 0.48
MKNK2 Q9HBH9 1/20 0.48
PARP1 P09874 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14334921 0.84 MKNK1 (0.54) ROCK2MKNK1MKNK2
SCHEMBL23458839 0.84 ROCK2 (0.53) ROCK2MKNK1MKNK2
SCHEMBL29882509 0.81 CHRNB2 (0.48) IRAK4CHEK1KCNH2CHRNB2CHRNA4
SCHEMBL14334551 0.81 IRAK4 (0.59) IRAK4CHRNB2CHRNA4ROCK2PARP1
SCHEMBL14334257 0.80 CHRNB2 (0.55) IRAK4CHEK1KCNH2CHRNB2CHRNA4
SCHEMBL16759169 0.79 KCNH2 (0.53) IRAK4CHEK1KCNH2CHRNB2CHRNA4
SCHEMBL20646781 0.78 RAB9A (0.48) ROCK2
SCHEMBL20646783 0.78 RAB9A (0.48) ROCK2
SCHEMBL3675210 0.78 ROCK2 (0.47) ROCK2
SCHEMBL6012159 0.76 ROCK2 (0.49) ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012176123-A1 3 - IMIDAZOLYL- INDOLES FOR THE TREATMENT OF PROLIFERATIVE DISEASES NOVARTIS AG (CH) 2012-12-27 WO disclosed