Tenofovir Diphosphate

Tenofovir Diphosphate

SCHEMBL14354588

C[C@H](Cn1cnc2c(N)ncnc21)OCP(=O)(O)OP(=O)(O)OP(=O)(O)O

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 16/20 0.77
CYP2D6 P10635 15/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tenofovir Diphosphate SCHEMBL29395812 1.00 CYP3A4 (0.77) CYP3A4CYP2D6
Tenofovir Diphosphate SCHEMBL29466912 1.00 CYP3A4 (0.77) CYP3A4CYP2D6
Tenofovir Diphosphate SCHEMBL24809661 1.00 CYP3A4 (0.77) CYP3A4CYP2D6
SCHEMBL14440381 0.96 CYP3A4 (0.80) CYP3A4CYP2D6
SCHEMBL24809662 0.96 CYP3A4 (0.80) CYP3A4CYP2D6
SCHEMBL19600198 0.94 CYP3A4 (0.77) CYP3A4CYP2D6
SCHEMBL20313254 0.92 CYP3A4 (0.74) CYP3A4CYP2D6
SCHEMBL13394187 0.91 CYP3A4 (0.75) CYP3A4CYP2D6
SCHEMBL20321881 0.90 CYP3A4 (0.71) CYP3A4CYP2D6
Tenofovir Anhydrous SCHEMBL400717 0.89 CYP3A4 (0.91) CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3334743-B1 ANTIVIRAL BETA-AMINO ACID ESTER PHOSPHODIAMIDE COMPOUNDS MERCK SHARP & DOHME LLC (US) 2023-11-29 EP disclosed
US-11826375-B2 Phosphinic amide prodrugs of tenofovir MERCK SHARP & DOHME LLC (US) 2023-11-28 US disclosed
US-11826375-B2 Phosphinic amide prodrugs of tenofovir MERCK SHARP & DOHME LLC (US) 2023-11-28 US disclosed
EP-3386512-B1 ANTIVIRAL PHOSPHODIAMIDE PRODRUGS OF TENOFOVIR MERCK SHARP & DOHME LLC (US) 2023-11-22 EP disclosed
WO-2022271880-A1 METHODS OF TREATING MEDICAL CONDITIONS AND INHIBITING LINE1 REVERSE TRANSCRIPTASE USING A SUBSTITUTED ADENINYL-PROPYLOXY PHOSPHONIC ACID OR RELATED COMPOUND ROME THERAPEUTICS, INC. (US) 2022-12-29 WO disclosed
EP-3559011-B1 ANTIVIRAL ESTER PRODRUGS OF TENOFOVIR MERCK SHARP & DOHME (US) 2022-04-13 EP disclosed
US-11123355-B2 Antiviral benzyl-amine phosphodiamide compounds IDENIX PHARMACEUTICALS LLC (US) 2021-09-21 US disclosed
EP-3390413-B1 ANTIVIRAL OXIME PHOSPHORAMIDE COMPOUNDS MERCK SHARP & DOHME (US) 2020-08-19 EP disclosed
US-10745428-B2 Antiviral phosphodiamide prodrugs of tenofovir IDENIX PHARMACEUTICALS LLC (US) 2020-08-18 US disclosed
US-10736908-B2 Antiviral aryl-amide phosphodiamide compounds MERCK SHARP & DOHME CORP. (US) 2020-08-11 US disclosed
US-20150315221-A1 NUCLEOSIDE KINASE BYPASS COMPOSITIONS AND METHODS MERCK SHARP & DOHME CORP. (US) 2015-11-05 US disclosed
EP-2579871-B1 TOPICAL ANTIVIRAL FORMULATIONS FOR PREVENTION OF TRANSMISSION OF HSV-2 GILEAD SCIENCES INC (US) 2015-08-26 EP disclosed
WO-2014088923-A1 NUCLEOSIDE KINASE BYPASS COMPOSITIONS AND METHODS MERCK SHARP & DOHME CORP. (US) 2014-06-12 WO disclosed
US-20130216590-A1 TOPICAL ANTIVIRAL FORMULATIONS FOR PREVENTION OF TRANSMISSION OF HSV-2 GILEAD SCIENCES, INC. 2013-08-22 US disclosed
US-20130216590-A1 TOPICAL ANTIVIRAL FORMULATIONS FOR PREVENTION OF TRANSMISSION OF HSV-2 GILEAD SCIENCES, INC. 2013-08-22 US disclosed
US-20130216590-A1 TOPICAL ANTIVIRAL FORMULATIONS FOR PREVENTION OF TRANSMISSION OF HSV-2 GILEAD SCIENCES, INC. 2013-08-22 US disclosed
EP-2579871-A1 TOPICAL ANTIVIRAL FORMULATIONS FOR PREVENTION OF TRANSMISSION OF HSV-2 Gilead Sciences, Inc. (US) 2013-04-17 EP disclosed
US-20070281911-A1 Use of Adefovir or Tenofovir for Inhibiting Mmtv-Like Viruses Involved in Breast Cancer and Primary Biliary Cirrhosis GILEAD SCIENCES INC. (US) 2007-12-06 US disclosed
US-20070190523-A1 Method and compositions for identifying anti-hiv therapeutic compounds GILEAD SCIENCES, INC. 2007-08-16 US disclosed
US-20070190523-A1 Method and compositions for identifying anti-hiv therapeutic compounds GILEAD SCIENCES, INC. 2007-08-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10736908-B2 Antiviral aryl-amide phosphodiamide compounds PNP, TYMP, DUT CYP3A4 1082/4885CYP2D6 1883/4885
US-11123355-B2 Antiviral benzyl-amine phosphodiamide compounds TYMP, PNP, POLI CYP3A4 2278/4885CYP2D6 3727/4885
US-20150315221-A1 NUCLEOSIDE KINASE BYPASS COMPOSITIONS AND METHODS DCK, DTYMK, TK1 CYP3A4 1852/4885CYP2D6 1377/4885
US-10745428-B2 Antiviral phosphodiamide prodrugs of tenofovir PNP, TYMP, PPA1 CYP3A4 628/4885CYP2D6 1334/4885
US-20130216590-A1 TOPICAL ANTIVIRAL FORMULATIONS FOR PREVENTION OF TRANSMISSION OF HSV-2 PRPH, TK1, PLP2 CYP3A4 4002/4885CYP2D6 1734/4885
US-11826375-B2 Phosphinic amide prodrugs of tenofovir TYMP, PPA1, PNP CYP3A4 1743/4885CYP2D6 2129/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.