SCHEMBL14367145

SCHEMBL14367145

COc1ccc(-c2ccc(/C=C/C(C)=O)cc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 3/20 0.71
HDAC6 Q9UBN7 3/20 0.71
HDAC3 O15379 2/20 0.71
HDAC1 Q13547 2/20 0.71
HDAC2 Q92769 2/20 0.71
HDAC4 P56524 1/20 0.71
HDAC7 Q8WUI4 1/20 0.71
HDAC10 Q969S8 1/20 0.71
HDAC11 Q96DB2 1/20 0.71
HDAC9 Q9UKV0 1/20 0.71
HDAC5 Q9UQL6 1/20 0.71
F3 P13726 3/20 0.68
THRB P10828 1/20 0.66
ATM Q13315 1/20 0.66
GSK3B P49841 2/20 0.64
BACE1 P56817 1/20 0.58
BCHE P06276 1/20 0.57
CYP3A4 P08684 1/20 0.57
NFKB1 P19838 1/20 0.57
NFKB2 Q00653 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL872009 0.94 F3 (0.75) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL872010 0.94 F3 (0.75) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL26124951 0.94 F3 (0.75) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL7967986 0.86 THRB (0.89) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL12473720 0.86 THRB (0.89) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL7967988 0.86 THRB (0.89) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL13067871 0.84 HDAC8 (0.69) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL8267192 0.84 HDAC8 (0.73) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL22490432 0.84 KMT2A (0.69) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL3292542 0.83 HDAC8 (1.00) HDAC8HDAC6HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7291743-B2 Isoxazole derivatives and methods of treating nitric oxide mediated diseases GENEBLUE CORPORATION (US) 2007-11-06 US disclosed