SCHEMBL14386157

SCHEMBL14386157

CN(C)C/C=C1\CC(N2CCC(Cc3ccc(Br)cc3Cl)C2=O)CCC1=O

nearest known ligand 0.31

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.31
METAP1 P53582 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12432115 0.89 PYCR1 (0.32) HSD11B1
SCHEMBL14386160 0.89 OPRM1 (0.35) HSD11B1METAP1
SCHEMBL12432125 0.81 OPRM1 (0.33) HSD11B1
SCHEMBL12432116 0.80 P2RX7 (0.33) HSD11B1METAP1
SCHEMBL14386159 0.79 HSD11B1 (0.32) HSD11B1
SCHEMBL12432106 0.79 P2RX7 (0.36)
SCHEMBL2208101 0.78 HSD11B1 (0.41) HSD11B1
SCHEMBL12432112 0.78 OPRM1 (0.36) HSD11B1METAP1
SCHEMBL2990822 0.75 HSD11B1 (0.54) HSD11B1
SCHEMBL474663 0.74 HSD11B1 (0.41) HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007124254-A2 CYCLOHEXYLPYRAZOLE-LACTAM DERIVATIVES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE 1 ELI LILLY AND COMPANY (US) 2007-11-01 WO disclosed