SCHEMBL14398136

SCHEMBL14398136

O=Cc1sccc1-c1c(C(=O)O)ccc2ccccc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 1/20 0.61
LDHA P00338 1/20 0.47
SOS1 Q07889 1/20 0.45
NR4A1 P22736 1/20 0.44
NR4A2 P43354 1/20 0.44
NR4A3 Q92570 1/20 0.44
ERN1 O75460 1/20 0.41
ALDH1A1 P00352 3/20 0.40
HPGD P15428 3/20 0.40
LMNA P02545 1/20 0.40
MCL1 Q07820 1/20 0.40
ACMSD Q8TDX5 1/20 0.40
CDC25B P30305 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
KDM4E B2RXH2 2/20 0.39
RORC P51449 1/20 0.39
RORB Q92753 1/20 0.39
PTPN1 P18031 1/20 0.39
CSNK2A2 P19784 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14398126 0.81 WDR5 (0.58) WDR5LDHASOS1NR4A1NR4A2
SCHEMBL31134224 0.80 ERN1 (0.41) WDR5ERN1ALDH1A1HPGDMEN1
SCHEMBL895573 0.78 WDR5 (1.00) WDR5LDHASOS1NR4A1NR4A2
SCHEMBL29721418 0.78 WDR5 (1.00) WDR5LDHASOS1NR4A1NR4A2
SCHEMBL14398058 0.77 KDM4E (0.46) ERN1ALDH1A1HPGDLMNAKMT2A
SCHEMBL14398192 0.75 MYC (0.51) NR4A1ALDH1A1HPGDLMNAMCL1
SCHEMBL967386 0.75 RORC (0.47) ERN1ALDH1A1MCL1ACMSDMEN1
SCHEMBL29458346 0.75 WDR5 (0.79) WDR5LDHASOS1NR4A1NR4A2
SCHEMBL9124028 0.75 WDR5 (0.79) WDR5LDHASOS1NR4A1NR4A2
SCHEMBL8595668 0.73 WDR5 (0.76) WDR5LDHASOS1NR4A1NR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007117180-A1 AZAHETEROCYCLES, COMBINATORY LIBRARY, FOCUSED LIBRARY, PHARMACEUTICAL COMPOSITION AND METHODS FOR THE PRODUCTION THEREOF 'CHEMICAL DIVERSITY RESEARCH INSTITUTE' LTD. (RU) 2007-10-18 WO disclosed