SCHEMBL1440863

SCHEMBL1440863

CC(C)COC(=O)N1CC(C=O)C1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.42
TSHR P16473 3/20 0.39
HDAC2 Q92769 1/20 0.38
KIT P10721 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37
P2RX4 Q99571 1/20 0.36
MEN1 O00255 1/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 1/20 0.35
KCNK3 O14649 1/20 0.35
KCNK9 Q9NPC2 1/20 0.35
HSD11B1 P28845 1/20 0.34
POLB P06746 1/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3830772 0.87 RAB9A (0.44) RAB9ATSHRKITMEN1HPGD
SCHEMBL5782598 0.85 RAB9A (0.49) RAB9ATSHRKITMEN1HPGD
SCHEMBL1440841 0.83 RAB9A (0.47) RAB9ATSHRKITMEN1HPGD
SCHEMBL14243062 0.80 CHRNB2 (0.54) RAB9ATSHRHDAC2KITCHRNB2
SCHEMBL1692767 0.80 RAB9A (0.45) RAB9ATSHRHDAC2KITCHRNB2
SCHEMBL2229068 0.79 RAB9A (0.44) RAB9ATSHRHDAC2KITCHRNB2
SCHEMBL19308678 0.79 HDAC2 (0.44) RAB9ATSHRHDAC2KITCHRNB2
SCHEMBL15703162 0.77 RAB9A (0.43) RAB9ATSHRHDAC2KITCHRNB2
SCHEMBL5568829 0.77 RAB9A (0.43) RAB9ATSHRHDAC2KITCHRNB2
SCHEMBL20002117 0.77 RAB9A (0.43) RAB9ATSHRHDAC2KITCHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2473056-A1 CHEMICAL COMPOUNDS GlaxoSmithKline LLC (US) 2012-07-11 EP disclosed
WO-2011028596-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2011-03-10 WO disclosed
WO-1997042189-A1 AZETIDINE, PYRROLIDINE AND PIPERIDINE DERIVATIVES AS 5-HT RECEPTOR AGONISTS MERCK SHARP & DOHME LIMITED (GB) 1997-11-13 WO disclosed