SCHEMBL14422651

SCHEMBL14422651

FC(F)(F)c1ccccc1-c1nnc2ccc(NC3CC3)nn12

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 13/20 0.64
FLT3 P36888 2/20 0.57
GSK3B P49841 2/20 0.57
JAK2 O60674 1/20 0.57
CDK2 P24941 1/20 0.57
JAK3 P52333 1/20 0.57
PRKCQ Q04759 1/20 0.57
IRAK4 Q9NWZ3 1/20 0.57
AURKA O14965 1/20 0.54
MALT1 Q9UDY8 6/20 0.52
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
KCNH2 Q12809 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14422661 0.84 PIM1 (0.68) PIM1FLT3GSK3BJAK2CDK2
SCHEMBL14422682 0.79 PIM1 (0.64) PIM1FLT3GSK3BJAK2CDK2
SCHEMBL14422647 0.78 PIM1 (1.00) PIM1FLT3GSK3BJAK2CDK2
SCHEMBL14422627 0.78 PIM1 (1.00) PIM1FLT3GSK3BJAK2CDK2
SCHEMBL14422660 0.77 PIM1 (1.00) PIM1FLT3GSK3BJAK2CDK2
SCHEMBL14422673 0.76 PIM1 (0.44) PIM1FLT3GSK3B
SCHEMBL29767394 0.76 ALDH1A1 (0.55)
SCHEMBL14422683 0.75 HSD11B1 (0.41) PIM1FLT3GSK3B
SCHEMBL14422668 0.74 PIM1 (1.00) PIM1FLT3GSK3BJAK2CDK2
SCHEMBL14422677 0.73 PIM1 (1.00) PIM1FLT3GSK3BJAK2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7268136-B2 Compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-09-11 US disclosed