Flomoxef

Flomoxef

SCHEMBL14423926

CO[C@@]1(NC(=O)CSC(F)F)C(=O)N2C(C(=O)O)=C(CSc3nnnn3CCO)COC21

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Flomoxef. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.57
CMA1 P23946 18/20 0.54
HSD17B10 Q99714 1/20 0.49
TDP1 Q9NUW8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Flomoxef SCHEMBL49438 1.00 PTGS1 (0.57) PTGS1CMA1HSD17B10TDP1
Flomoxef SCHEMBL65125 0.99 PTGS1 (0.57) PTGS1CMA1HSD17B10TDP1
Flomoxef SCHEMBL27661462 0.99 PTGS1 (0.57) PTGS1CMA1HSD17B10TDP1
Flomoxef SCHEMBL30531854 0.93 HSD17B10 (0.58) PTGS1CMA1HSD17B10TDP1
Flomoxef SCHEMBL30716855 0.93 HSD17B10 (0.58) PTGS1CMA1HSD17B10TDP1
Flomoxef SCHEMBL27896310 0.92 PTGS1 (0.51) PTGS1CMA1HSD17B10TDP1
SCHEMBL30515648 0.86 CMA1 (0.60) PTGS1CMA1
Flomoxef SCHEMBL30515667 0.82 PTGS1 (0.44) PTGS1CMA1HSD17B10TDP1
Flomoxef SCHEMBL18065040 0.78 NR1I2 (0.58) PTGS1HSD17B10TDP1
Flomoxef SCHEMBL2563269 0.78 ABCB11 (0.53) PTGS1CMA1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007105253-A2 PREPARATION OF (1-OXA- OR l-THIA-)3- CEPHEM DERIVATIVES CARTHESIA S.A.S. DI EMANUELA MIGLIAVACCA & C. (IT) 2007-09-20 WO disclosed