SCHEMBL14433474

SCHEMBL14433474

CN(CCNc1cccnc1N)S(C)(=O)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 5/20 0.46
SLC40A1 Q9NP59 2/20 0.40
SHMT2 P34897 1/20 0.39
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38
GLO1 Q04760 1/20 0.38
PIK3CD O00329 1/20 0.38
CYP2C19 P33261 1/20 0.37
HRH3 Q9Y5N1 1/20 0.35
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
PTK2 Q05397 3/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
NCF1 P14598 1/20 0.34
KAT2B Q92831 1/20 0.34
MEN1 O00255 1/20 0.33
NFKBIA P25963 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5258796 0.80 SLC40A1 (0.36) SLC40A1ALOX15HTTGLO1CYP2C19
SCHEMBL14433127 0.79 HTR5A (0.48) BACE1SLC40A1SHMT2ALOX15HTT
SCHEMBL9977915 0.78 BACE1 (0.49) BACE1SLC40A1SHMT2ALOX15HTT
SCHEMBL5255932 0.78 L3MBTL1 (0.43) SLC40A1ALOX15HTTGLO1PIK3CD
SCHEMBL19897481 0.71 BACE1 (0.54) BACE1SHMT2NOS3NOS1NOS2
SCHEMBL9689711 0.71 BACE1 (0.57) BACE1SHMT2CYP2C19HSP90AA1HSP90AB1
SCHEMBL4823208 0.70 L3MBTL1 (0.41) PIK3CDCYP2C19NCF1MEN1KMT2A
SCHEMBL3060454 0.70 BACE1 (0.61) BACE1SHMT2NOS3NOS1NOS2
SCHEMBL4711248 0.70 BACE1 (0.53) BACE1SHMT2HSP90AA1HSP90AB1NOS3
SCHEMBL9977955 0.70 BACE1 (0.53) BACE1SHMT2HTTCYP2C19HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1467970-B1 HYDROXYNAPHTHYRIDINONE CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2007-08-22 EP disclosed