SCHEMBL14439831

SCHEMBL14439831

CC(C)c1nc(COCc2ccccc2)n(CCCO)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
VCP P55072 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
RHEB Q15382 1/20 0.32
HSP90B1 P14625 2/20 0.32
TRAP1 Q12931 2/20 0.32
SLC5A2 P31639 1/20 0.31
TSHR P16473 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
GRM5 P41594 3/20 0.31
ADAMTS5 Q9UNA0 2/20 0.31
MMP2 P08253 1/20 0.31
MMP13 P45452 1/20 0.31
ADAM17 P78536 1/20 0.31
DHODH Q02127 1/20 0.31
HSP90AA1 P07900 1/20 0.30
HSP90AB1 P08238 1/20 0.30
TP53 P04637 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8109133 0.94 VCP (0.35) HDAC1HDAC8VCPTDP1RHEB
SCHEMBL6972304 0.91 HSP90B1 (0.37) HDAC1HDAC8VCPTDP1HSP90B1
SCHEMBL14439829 0.90 VCP (0.36) HDAC1HDAC8VCPTDP1RHEB
SCHEMBL6972409 0.89 VCP (0.35) VCPTDP1SLC5A2DHODHTP53
SCHEMBL6965896 0.88 VCP (0.36) HDAC1HDAC8VCPTDP1SLC5A2
SCHEMBL14439828 0.88 TDP1 (0.40) VCPTDP1SLC5A2TSHRDHODH
SCHEMBL6966496 0.87 VCP (0.37) VCPTDP1SLC5A2TSHRADAMTS5
SCHEMBL6973959 0.87 VCP (0.35) VCPTDP1SLC5A2ADAMTS5MMP2
SCHEMBL14439841 0.86 VCP (0.36) VCPTDP1SLC5A2TSHRADAMTS5
SCHEMBL6960981 0.86 TLR8 (0.33) TDP1RHEB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070190523-A1 Method and compositions for identifying anti-hiv therapeutic compounds GILEAD SCIENCES, INC. 2007-08-16 US disclosed