SCHEMBL14448263

SCHEMBL14448263

O=C(Nc1ccc2nccnc2c1)C1CN2CCC1CC2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 11/20 0.47
ALDH1A1 P00352 9/20 0.47
HPGD P15428 7/20 0.47
HSD17B10 Q99714 4/20 0.47
MAPT P10636 4/20 0.47
KMT2A Q03164 4/20 0.47
CASP1 P29466 3/20 0.47
GAA P10253 3/20 0.47
TP53 P04637 3/20 0.47
CASP7 P55210 2/20 0.47
MAPK1 P28482 1/20 0.45
NPC1 O15118 6/20 0.45
RAB9A P51151 6/20 0.45
SMN1; SMN2 Q16637 5/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
NFKB1 P19838 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5483889 0.99 KDM4E (0.46) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL14448258 0.85 HTR3A (0.58) MAPTKMT2ANPC1RAB9AMEN1
Hydrochloric Acid SCHEMBL5467852 0.84 HTR3A (0.57) MAPTKMT2ANPC1RAB9AMEN1
SCHEMBL259751 0.81 CHRM5 (0.56)
SCHEMBL263699 0.81 CHRM5 (0.56)
SCHEMBL263519 0.81 CHRM5 (0.58)
SCHEMBL263703 0.77 ALDH1A1 (0.37) ALDH1A1MAPTGAANPC1RAB9A
SCHEMBL14448261 0.76 CYP1A2 (0.53) KDM4EALDH1A1HPGDMAPTKMT2A
Hydrochloric Acid SCHEMBL5471928 0.75 CYP1A2 (0.52) KDM4EALDH1A1HPGDMAPTKMT2A
SCHEMBL6556747 0.75 CHRNA7 (0.62) ALDH1A1TP53NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7247728-B2 Bicyclic N-arylamides BAYER HEALTHCARE AG (DE) 2007-07-24 US disclosed
US-7247728-B2 Bicyclic N-arylamides BAYER HEALTHCARE AG (DE) 2007-07-24 US disclosed