SCHEMBL1444909

SCHEMBL1444909

O=C(O)C1C=Nc2ccccc2C1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.38
HTT P42858 2/20 0.38
HBB P68871 2/20 0.38
ALOX15 P16050 1/20 0.38
EDNRB P24530 1/20 0.36
EDNRA P25101 1/20 0.36
THRB P10828 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ADORA3 P0DMS8 1/20 0.35
CHRM1 P11229 1/20 0.35
TBXA2R P21731 1/20 0.35
PTGS1 P23219 1/20 0.35
ADRA1A P35348 1/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27338358 0.98 MAPT (0.37) MAPTHTTHBBALOX15EDNRB
SCHEMBL2934359 0.86 MAPT (0.40) MAPTHTTHBBALOX15THRB
SCHEMBL1450636 0.84 GABRP (0.34) MAPTHTTHBBALOX15THRB
SCHEMBL28846735 0.80 GABRP (0.35) MAPTHTTHBBALOX15GABRP
SCHEMBL28628608 0.78 LMNA (0.30) EDNRBEDNRAGABRPGABRDGABRA1
SCHEMBL6778036 0.78 NPSR1 (0.35) MAPTTHRBMEN1KMT2AALDH1A1
SCHEMBL17320675 0.76 LMNA (0.46) MAPTEDNRBEDNRAMEN1KMT2A
SCHEMBL2933046 0.76 GABRP (0.37) MAPTHTTHBBALOX15MEN1
SCHEMBL5566400 0.75 KMT2A (0.35) MAPTHTTHBBALOX15THRB
SCHEMBL9615419 0.75 NPSR1 (0.44) MAPTMEN1KMT2ALMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 320 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118067873-A Method for detecting impurities in moxifloxacin hydrochloride sodium chloride injection 华夏生生药业(北京)有限公司 2024-05-24 CN claimed
CN-116606280-A Fluoroquinolone compound and application thereof in preparation of antibacterial drugs 广东工业大学 2023-08-18 CN claimed
CN-114539213-A Fluoroquinolone compound and preparation method and application thereof 广东工业大学 2022-05-27 CN claimed
EP-2398919-B1 METHOD FOR IDENTIFYING A SUBPOPULATION OF MAMMALIAN CELLS WITH DISTINCTIVE RIBOSOME TRANSLATION PROFILES UNIV WAYNE STATE (US) 2018-07-25 EP claimed
US-9388405-B2 Method for identifying a subpopulation of mammalian cells with distinctive ribosome translation profiles WAYNE STATE UNIVERSITY (US) 2016-07-12 US claimed
EP-1401829-B1 NOVEL HETEROCYCLIC ANTIBACTERIAL COMPOUNDS MICROBIOTIX INC (US) 2012-08-22 EP claimed
US-20120107828-A1 METHOD FOR IDENTIFYING A SUBPOPULATION OF MAMMALIAN CELLS WITH DISTINCTIVE RIBOSOME TRANSLATION PROFILES WAYNE STATE UNIVERSITY (US) 2012-05-03 US claimed
CN-102276528-A Chemical preparation method of sarafloxacin hydrochloride XINCHANG HEBAO BIOLOG TECHNOLOGY CO LTD 2011-12-14 CN claimed
JP-4669607-B2 2011-04-13 JP claimed
WO-2010096594-A2 METHOD FOR IDENTIFYING A SUBPOPULATION OF MAMMALIAN CELLS WITH DISTINCTIVE RIBOSOME TRANSLATION PROFILES WAYNE STATE UNIVERSITY (US) 2010-08-26 WO claimed
EP-0610958-A2 Intermediates in the preparation of 4-oxoquinoline-3-carboxylic acid derivatives UBE INDUSTRIES, LTD. (JP) 1994-08-17 EP claimed
WO-1993024481-A1 7-SUBSTITUTED-6-FLUORO-1,4-DIHYDRO-4-OXO-QUINOLINE-3-CARBOXYLIC ACID COMPOUNDS AND RELATED COMPOUNDS AS ANTIBACTERIAL AGENTS SYNPHAR LABORATORIES, INC. (CA) 1993-12-09 WO claimed
US-5237060-A Cyclization; amination BAYER AKTIENGESELLSCHAFT (DE) 1993-08-17 US claimed
EP-0253235-B1 1,8-BRIDGED 4-QUINOLONE CARBOXYLIC ACIDS AND MEDICAMENTS CONTANING THEM BAYER AG (DE) 1991-01-02 EP claimed
US-4859773-A Preparation of 1,8-bridged 4-quinoline-3-carboxylic acids BAYER AKTIENGESELLSCHAFT (DE) 1989-08-22 US claimed
US-4847375-A Antibacterial 1,8-bridged 4-quinoline-3-carboxylic acids BAYER AKTIENGESELLSCHAFT (DE) 1989-07-11 US claimed
US-4816451-A Antibacterial 1,8-bridged 4-quinolonecarboxylic acids BAYER AKTIENGESELLSCHAFT (DE) 1989-03-28 US claimed
US-4725595-A 1,8-bridged 4-quinolone-3-carboxylic acid antibacterials BAYER AKTIENGESELLSCHAFT (DE) 1988-02-16 US claimed
CN-86104256-A 1, the preparation method of 8-bridging 4-quinolone-3-carboxylic-acid 1987-03-18 CN claimed
EP-0179239-A2 7-(Pyridinyl)-/-alkyl-1,4-dihydro-4-oxo-3-quinolinecarboxylic acid having antibacterial activity and preparation thereof STERLING DRUG INC. (US) 1986-04-30 EP claimed