SCHEMBL14469683

SCHEMBL14469683

CC1(C)C=C(C(=O)OCc2ccccc2)c2cc(F)c(Cl)cc2OC1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.40
PKM P14618 1/20 0.39
ADORA2B P29275 1/20 0.37
AKR1B1 P15121 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
SLC6A2 P23975 1/20 0.35
SLC6A3 Q01959 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
NOTUM Q6P988 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14469812 0.92 KMT2A (0.38) GPBAR1PKMADORA2BAKR1B1KMT2A
SCHEMBL14469705 0.82 TDP1 (0.42) PKMADORA2BKMT2ASLC6A2SLC6A3
SCHEMBL14469684 0.81 PRKCZ (0.42) KMT2ASLC6A2SLC6A3TDP1TSHR
SCHEMBL14469714 0.80 TSHR (0.45) GPBAR1KMT2ASLC6A2SLC6A3TDP1
SCHEMBL14469745 0.80 ALDH1A1 (0.43) GPBAR1PKMKMT2AMEN1SLC6A2
SCHEMBL20830732 0.66 TDP1 (0.58) KMT2AMEN1SLC6A2SLC6A3TDP1
SCHEMBL24117922 0.64 TDP1 (0.54) KMT2ASLC6A2SLC6A3TDP1TSHR
SCHEMBL22245235 0.63 TDP1 (0.54) GPBAR1KMT2ASLC6A2SLC6A3TDP1
SCHEMBL25910700 0.63 TDP1 (0.46) GPBAR1PKMKMT2ASLC6A2SLC6A3
SCHEMBL31448243 0.63 ALDH1A1 (0.50) PKMKMT2ASLC6A2SLC6A3TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1686983-B1 USE OF PENTADIENOIC ACID DERIVATES FOR TREATEMENT OF HYPERURICEMIA MERCK PATENT GMBH (DE) 2007-07-11 EP disclosed