SCHEMBL14486197

SCHEMBL14486197

COc1cccc(S(=O)(=O)c2ccc(S(=O)(=O)c3cccc(OC)c3)c3cnccc23)c1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 9/20 0.52
GAA P10253 1/20 0.51
CYP11B1 P15538 2/20 0.46
CYP11B2 P19099 2/20 0.46
NAMPT P43490 1/20 0.45
FEN1 P39748 1/20 0.45
SLC22A12 Q96S37 1/20 0.43
MGAT2 Q10469 1/20 0.43
KEAP1 Q14145 1/20 0.43
PTGS1 P23219 1/20 0.43
MTNR1B P49286 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14485855 0.83 PKM (0.53) NFE2L2GAANAMPTKEAP1PTGS1
SCHEMBL31352975 0.75 MTNR1B (0.56) NFE2L2KEAP1MTNR1BALDH1A1
SCHEMBL3151230 0.75 MTNR1B (0.56) NFE2L2KEAP1MTNR1BALDH1A1
SCHEMBL3888075 0.75 HTR6 (0.51) NFE2L2GAA
SCHEMBL3885920 0.74 HTR6 (0.54) NFE2L2GAACYP11B1CYP11B2NAMPT
SCHEMBL3899853 0.73 HASPIN (0.46) NFE2L2GAA
SCHEMBL14486062 0.72 COMT (0.50) GAAALDH1A1
SCHEMBL17615769 0.72 NFE2L2 (0.43) NFE2L2GAACYP11B1CYP11B2NAMPT
SCHEMBL14486083 0.71 NAMPT (0.44) NAMPTALDH1A1
SCHEMBL28499568 0.71 NFE2L2 (0.47) NFE2L2GAAFEN1KEAP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013005157-A1 SULFONE DERIVATIVES AND THEIR USE AS PKM2 MODULATORS FOR THE TREATMENT OF CANCER LUPIN LIMITED (IN) 2013-01-10 WO disclosed