SCHEMBL14498482

SCHEMBL14498482

Cc1cc2[nH]c(=O)oc(=O)c2s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 5/20 0.41
NOS2 P35228 4/20 0.41
NOS3 P29474 3/20 0.41
F2 P00734 1/20 0.39
CFD P00746 1/20 0.39
KMO O15229 1/20 0.35
PDGFRA P16234 1/20 0.35
MAPK8 P45983 1/20 0.35
CDK5 Q00535 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
MAOA P21397 3/20 0.35
MAOB P27338 3/20 0.35
OGT O15294 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
ADRA2A P08913 1/20 0.33
TSHR P16473 1/20 0.33
THPO P40225 1/20 0.33
BLM P54132 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3548193 0.79 ERCC5 (0.53) NOS1NOS2NOS3F2CFD
SCHEMBL25541170 0.77 NOS1 (0.43) NOS1NOS2NOS3F2CFD
SCHEMBL14403068 0.75 F2 (0.34) NOS1NOS2NOS3F2CFD
SCHEMBL13392528 0.73 PKM (0.33) NPSR1PKMPKLR
SCHEMBL1523074 0.71 ERCC5 (0.54) NOS1F2CFDPDGFRAMAPK8
SCHEMBL3932932 0.70 F2 (0.39) NOS1NOS2NOS3F2CFD
SCHEMBL4214560 0.69 CDC7 (0.51) PKMPKLRERCC5FEN1
SCHEMBL19427807 0.67 ALDH1A1 (0.37) PKMPKLR
SCHEMBL27398191 0.66 ADORA2B (0.43) LMNATSHRBLMPKMPKLR
SCHEMBL10618031 0.65 F2 (0.50) NOS1NOS2NOS3F2CFD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7235566-B2 Pyridinone derivatives for treatment of atherosclerosis SMITHKLINE BEECHAM P.L.C. (GB) 2007-06-26 US disclosed
US-7235566-B2 Pyridinone derivatives for treatment of atherosclerosis SMITHKLINE BEECHAM P.L.C. (GB) 2007-06-26 US disclosed