SCHEMBL14503548

SCHEMBL14503548

CC(=O)N1CCN(c2nc(Nc3ccc(NC(=O)c4ccc(C)cc4)c(O)c3)nc(N3CCCCC3)n2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.53
MAPT P10636 6/20 0.50
ALDH1A1 P00352 2/20 0.50
CYP2C9 P11712 1/20 0.50
HPGD P15428 1/20 0.50
CYP2C19 P33261 1/20 0.50
SMN1; SMN2 Q16637 3/20 0.47
LMNA P02545 3/20 0.47
CTNNB1 P35222 2/20 0.45
TCF7L2 Q9NQB0 2/20 0.45
HTT P42858 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
NPC1 O15118 2/20 0.43
KDM4E B2RXH2 1/20 0.43
RAB9A P51151 1/20 0.43
MCL1 Q07820 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
GBA1 P04062 3/20 0.43
POLB P06746 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14503191 0.94 PTGS2 (0.57) PTGS2MAPTALDH1A1CYP2C9CYP2C19
SCHEMBL14503163 0.94 PTGS2 (0.57) PTGS2MAPTALDH1A1CYP2C9CYP2C19
SCHEMBL14503676 0.88 PTGS2 (0.52) PTGS2MAPTALDH1A1CYP2C9CYP2C19
SCHEMBL5380874 0.88 ALDH1A1 (0.46) PTGS2MAPTALDH1A1CYP2C9HPGD
SCHEMBL14503628 0.88 MAPT (0.49) PTGS2MAPTALDH1A1CYP2C9HPGD
SCHEMBL14503642 0.87 PTGS2 (0.53) PTGS2MAPTALDH1A1CYP2C9CYP2C19
SCHEMBL14503664 0.86 PTGS2 (0.49) PTGS2MAPTALDH1A1SMN1; SMN2LMNA
SCHEMBL14503398 0.86 LMNA (0.58) PTGS2MAPTSMN1; SMN2LMNAHTT
SCHEMBL14503227 0.85 PTGS2 (0.56) PTGS2MAPTALDH1A1HPGDSMN1; SMN2
SCHEMBL14503143 0.85 PTGS2 (0.56) PTGS2MAPTALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7223759-B2 Antibacterial 3,5-diaminopiperidine-substituted aromatic and heteroaromatic compounds ANADYS PHARMACEUTICALS, INC. (US) 2007-05-29 US disclosed
US-7223759-B2 Antibacterial 3,5-diaminopiperidine-substituted aromatic and heteroaromatic compounds ANADYS PHARMACEUTICALS, INC. (US) 2007-05-29 US disclosed