SCHEMBL14574

SCHEMBL14574

CC(C)(C)OC(=O)/N=C(/NCCCCN1CCC(n2cc3c(nc2=O)[nH]c2ccccc23)C1)NC(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.36
DRD3 P35462 3/20 0.35
FAAH O00519 2/20 0.35
ADRA2C P18825 1/20 0.35
CAMK2D Q13557 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HSD17B10 Q99714 1/20 0.34
SIGMAR1 Q99720 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14463 0.90 DRD2 (0.44) DRD2DRD3FAAHADRA2CCAMK2D
SCHEMBL14539 0.90 ADRA2C (0.36) DRD2DRD3FAAHADRA2CCAMK2D
SCHEMBL13698 0.79 DRD2 (0.37) DRD2DRD3KDM4EALDH1A1HSD17B10
SCHEMBL8076 0.79 DRD2 (0.37) DRD2DRD3KDM4EALDH1A1HSD17B10
SCHEMBL12062415 0.77 CHRM1 (0.48) DRD2KDM4EALDH1A1HSD17B10
SCHEMBL12061561 0.76 SLC6A4 (0.43)
SCHEMBL14551 0.73 ADRA1D (0.52) DRD2DRD3ALDH1A1SIGMAR1
SCHEMBL14077 0.72 SLC6A4 (0.47) DRD2DRD3
SCHEMBL7550 0.64 PDE5A (0.34) KDM4EALDH1A1HSD17B10SIGMAR1
SCHEMBL991815 0.64 TDP1 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011047319-A2 ANTIMICROBIAL COMPOUNDS AND METHODS OF MAKING AND USING THE SAME RIB-X PHARMACEUTICALS, INC. (US) 2011-04-21 WO disclosed