SCHEMBL14577909

SCHEMBL14577909

Cc1cc(C)c(C(=O)CCN2CCN(Cc3ccccc3)CC2)s1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.54
ALDH1A1 P00352 5/20 0.54
TSHR P16473 2/20 0.54
KMT2A Q03164 4/20 0.51
MEN1 O00255 2/20 0.50
HTR7 P34969 2/20 0.50
HTR1A P08908 2/20 0.50
MAPT P10636 1/20 0.47
POLB P06746 1/20 0.46
KDM4E B2RXH2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5353029 0.99 ACHE (0.53) ACHEALDH1A1TSHRKMT2AMEN1
Hydrochloric Acid SCHEMBL5357708 0.82 KMT2A (0.56) ALDH1A1KMT2AMEN1HTR1AKDM4E
Hydrochloric Acid SCHEMBL5373255 0.79 ALDH1A1 (0.62) ACHEALDH1A1TSHRKMT2AMEN1
SCHEMBL7980861 0.79 ACHE (0.53) ACHEALDH1A1TSHRKMT2AMEN1
SCHEMBL7984579 0.78 ACHE (0.52) ACHEALDH1A1TSHRKMT2AMEN1
Hydrochloric Acid SCHEMBL5364551 0.77 ACHE (0.51) ACHEALDH1A1TSHRKMT2AMEN1
SCHEMBL7970723 0.77 ACHE (0.51) ACHEALDH1A1TSHRKMT2AMEN1
Hydrochloric Acid SCHEMBL5360736 0.76 ACHE (0.50) ACHEALDH1A1TSHRKMT2AMEN1
SCHEMBL4512612 0.76 ALDH1A1 (0.71) ACHEALDH1A1KMT2AHTR7HTR1A
SCHEMBL5373264 0.76 ALDH1A1 (0.67) ACHEALDH1A1KMT2AHTR7HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7173132-B2 Certain substituted 1-aryl-3-piperazine-1′-yl propanones MOLECULAR GERIATRICS CORPORATION (US) 2007-02-06 US disclosed
US-7173132-B2 Certain substituted 1-aryl-3-piperazine-1′-yl propanones MOLECULAR GERIATRICS CORPORATION (US) 2007-02-06 US disclosed