SCHEMBL14587288

SCHEMBL14587288

CC(C)(C)OC(=O)N(C/C=C/Cl)c1ccccc1Br

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.37
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
NPC1 O15118 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
SSTR4 P31391 1/20 0.32
AKT1 P31749 1/20 0.32
RIPK1 Q13546 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
PAX8 Q06710 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14587285 0.85 KDM4E (0.33) AKT1L3MBTL1PAX8KDM4EALDH1A1
SCHEMBL3694335 0.84 LMNA (0.33) CYP3A4ALDH1A1
SCHEMBL3694334 0.84 LMNA (0.33) CYP3A4ALDH1A1
SCHEMBL3851116 0.81 SMN1; SMN2 (0.40) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL2400850 0.81 SMN1; SMN2 (0.40) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL2921603 0.79 NPSR1 (0.39) NPSR1MEN1KMT2ANPC1HTT
SCHEMBL13061313 0.76 HDAC1 (0.30) HDAC1HDAC8HDAC6
SCHEMBL2923486 0.75 SMN1; SMN2 (0.41) NPSR1MEN1KMT2ANPC1HTT
SCHEMBL31439848 0.75 ADRA2C (0.40) NPSR1MEN1KMT2ANPC1HTT
SCHEMBL15286185 0.74 NPSR1 (0.36) NPSR1MEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7179921-B2 Indoline and tetrahydro-quinolines as prodrugs for tumour treatment SCHOOL OF PHARMACY, UNIVERSITY OF LONDON (GB) 2007-02-20 US disclosed