SCHEMBL14587285

SCHEMBL14587285

CC(C)(C)OC(=O)N(CC=CCl)c1ccccc1I

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
AKT1 P31749 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.31
PAX8 Q06710 1/20 0.31
GSTO1 P78417 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14587288 0.85 NPSR1 (0.37) KDM4EALDH1A1AKT1L3MBTL1PAX8
SCHEMBL29009658 0.84 L3MBTL1 (0.38) KDM4EALDH1A1AKT1L3MBTL1GSTO1
SCHEMBL13061313 0.80 HDAC1 (0.30)
SCHEMBL5560364 0.79 ALDH1A1 (0.30) ALDH1A1
SCHEMBL3694334 0.79 LMNA (0.33) ALDH1A1
SCHEMBL3694335 0.79 LMNA (0.33) ALDH1A1
SCHEMBL29837260 0.79 HDAC3 (0.36) ALDH1A1AKT1L3MBTL1
SCHEMBL29837189 0.78 L3MBTL1 (0.41) AKT1L3MBTL1
SCHEMBL30758070 0.77 AKT1 (0.47) AKT1L3MBTL1
SCHEMBL5095964 0.77 BRD4 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7179921-B2 Indoline and tetrahydro-quinolines as prodrugs for tumour treatment SCHOOL OF PHARMACY, UNIVERSITY OF LONDON (GB) 2007-02-20 US disclosed