SCHEMBL14587747

SCHEMBL14587747

Cc1ccc(CNc2nc(NCCCN3CCCC3=O)nc3c2ncn3C(C)C)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 7/20 0.58
CCNB2 O95067 4/20 0.58
CCNB1 P14635 4/20 0.58
CCNB3 Q8WWL7 4/20 0.58
CDK2 P24941 10/20 0.56
TDP1 Q9NUW8 3/20 0.56
CCNE2 O96020 6/20 0.56
CCNE1 P24864 6/20 0.56
CCNA2 P20248 5/20 0.56
CCNA1 P78396 5/20 0.56
KDM4E B2RXH2 2/20 0.55
NPC1 O15118 2/20 0.55
MAPT P10636 2/20 0.55
CDK5 Q00535 3/20 0.54
CSNK1D P48730 1/20 0.54
CLK2 P49760 1/20 0.54
DYRK1A Q13627 1/20 0.54
HIPK4 Q8NE63 1/20 0.54
SRPK1 Q96SB4 1/20 0.54
CLK4 Q9HAZ1 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14587808 0.91 TDP1 (0.68) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL14587740 0.75 TDP1 (0.57) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL24669662 0.73 TDP1 (0.81) CDK1CCNB2CCNB1CCNB3CDK2
Bohemine SCHEMBL29572816 0.73 CDK1 (1.00) CDK1CCNB2CCNB1CCNB3CDK2
Bohemine SCHEMBL1443403 0.73 CDK1 (1.00) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL7112489 0.72 CDK1 (0.94) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL13497833 0.72 CDK5 (0.68) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL14587738 0.72 TDP1 (0.63) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL31069517 0.71 TDP1 (0.87) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL14587743 0.71 CDK1 (0.85) CDK1CCNB2CCNB1CCNB3CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176312-B2 Kinase inhibitor scaffolds and methods for their preparation THE SCRIPPS RESEARCH INSTITUTE (US) 2007-02-13 US disclosed