SCHEMBL1459622

SCHEMBL1459622

COS(=O)(=O)c1cccc2cccc(N)c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.40
RPS6KA3 P51812 1/20 0.40
MELK Q14680 1/20 0.40
STK24 Q9Y6E0 1/20 0.40
GAA P10253 2/20 0.39
F2 P00734 2/20 0.39
PRSS1 P07477 2/20 0.39
PRSS2 P07478 2/20 0.39
PRSS3 P35030 2/20 0.39
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
CA12 O43570 1/20 0.38
CYP2C9 P11712 1/20 0.38
CA4 P22748 1/20 0.38
CA6 P23280 1/20 0.38
CA5A P35218 1/20 0.38
CA7 P43166 1/20 0.38
CA14 Q9ULX7 1/20 0.38
CA5B Q9Y2D0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1459150 0.79 GAA (0.58) GAAF2CA1CA2CA9
SCHEMBL15172852 0.79 CA2 (0.61) JAK2RPS6KA3MELKSTK24GAA
SCHEMBL1458540 0.78 CA1 (0.43) JAK2RPS6KA3MELKSTK24GAA
Ammonia Solution, Strong SCHEMBL27361883 0.77 GAA (0.56) GAAF2CA1CA2CA9
SCHEMBL15274084 0.76 TTR (0.59) GAACA2TTRNSD2ALDH1A1
SCHEMBL179823 0.76 TTR (0.58) JAK2RPS6KA3MELKSTK24GAA
SCHEMBL29360969 0.76 TTR (0.58) JAK2RPS6KA3MELKSTK24GAA
SCHEMBL9098638 0.75 ALDH1A1 (0.44) JAK2RPS6KA3MELKSTK24GAA
Water SCHEMBL7765550 0.74 TTR (0.56) JAK2RPS6KA3MELKSTK24GAA
SCHEMBL21240726 0.74 TTR (0.56) JAK2RPS6KA3MELKSTK24GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130247309-A1 DYES AND BLENDS FOR SHADING DURING LAUNDRY BASF SE (DE) 2013-09-26 US disclosed
US-8178271-B2 Polymer having a sulfonic group or a sulfonate group and an amide group and method of producing same CANON KABUSHIKI KAISHA (JP) 2012-05-15 US disclosed
US-7935771-B2 Polymer having sulfonic acid group or sulfonic acid ester group and amide group, and toner for developing electrostatic latent image having the polymer CANON KABUSHIKI KAISHA (JP) 2011-05-03 US disclosed
EP-2292670-A2 Charge control agent, toner, image forming method, and image forming apparatus Canon Kabushiki Kaisha (JP) 2011-03-09 EP disclosed
US-20100233610-A1 POLYMER HAVING A SULFONIC GROUP OR A SULFONATE GROUP AND AN AMIDE GROUP AND METHOD OF PRODUCING SAME CANON KABUSHIKI KAISHA (JP) 2010-09-16 US disclosed
US-7795363-B2 Polymer having a sulfonic group or a sulfonate group and an amide group and method of producing same CANON KABUSHIKI KAISHA (JP) 2010-09-14 US disclosed
US-20100121023-A1 POLYMER HAVING A SULFONIC GROUP OR A SULFONATE GROUP AND AN AMIDE GROUP AND METHOD OF PRODUCING SAME CANON KABUSHIKI KAISHA (JP) 2010-05-13 US disclosed
EP-2184645-A2 Charge control agent, toner, image forming method and image forming apparatus Canon Kabushiki Kaisha (JP) 2010-05-12 EP disclosed
US-7638590-B2 Polyhydroxyalkanoate having amide, sulfonic acid or sulfonate ester group, charge control agent and toner CANON KABUSHIKI KAISHA (JP) 2009-12-29 US disclosed
US-7638194-B2 Developer carrying member, and developing assembly CANON KABUSHIKI KAISHA (JP) 2009-12-29 US disclosed
EP-1579277-B1 POLYHYDROXYALKANOATE CONTAINING AMIDE GROUP, SULFONIC GROUP, AND SULFONATE ESTER GROUP, METHOD FOR PRODUCING THE SAME, AND CHARGE CONTROL AGENT, TONER, IMAGE FORMING METHOD, AND IMAGE FORMING APPARATUS CANON KK (JP) 2006-09-06 EP disclosed
EP-1579276-B1 NOVEL POLYHYDROXYALKANOATE HAVING AMIDE, SULFONIC ACID OR SULFONATE ESTER GROUP, CHARGE CONTROL AGENT AND TONER CANON KK (JP) 2006-08-09 EP disclosed
US-20060035098-A1 Developer carrying member, and developing assembly CANON KABUSHIKI KAISHA (JP) 2006-02-16 US disclosed
US-20060014921-A1 Polyhydroxyalkanoate containing amide group, sulfonic group, and sulfonate ester group, method for producing the same, and charge control agent, toner, image forming method, and image forming apparatus CANON KABUSHIKI KAISHA (JP) 2006-01-19 US disclosed
US-20050287463-A1 Carrier for electrophotographic developer KANON KABUSHIKI KAISHA (JP) 2005-12-29 US disclosed
WO-2005108441-A2 POLYMER HAVING A SULFONIC GROUP OR A SULFONATE GROUP AND AN AMIDE GROUP AND METHOD OF PRODUCING SAME CANON KABUSHIKI KAISHA (JP) 2005-11-17 WO disclosed
EP-1579276-A1 NOVEL POLYHYDROXYALKANOATE HAVING AMIDE, SULFONIC ACID OR SULFONATE ESTER GROUP, CHARGE CONTROL AGENT AND TONER CANON KABUSHIKI KAISHA (JP) 2005-09-28 EP disclosed
EP-1579277-A1 POLYHYDROXYALKANOATE CONTAINING AMIDE GROUP, SULFONIC GROUP, AND SULFONATE ESTER GROUP, METHOD FOR PRODUCING THE SAME, AND CHARGE CONTROL AGENT, TONER, IMAGE FORMING METHOD, AND IMAGE FORMING APPARATUS Canon Kabushiki Kaisha (JP) 2005-09-28 EP disclosed
WO-2004061530-A1 POLYHYDROXYALKANOATE CONTAINING AMIDE GROUP, SULFONIC GROUP, AND SULFONATE ESTER GROUP, METHOD FOR PRODUCING THE SAME, AND CHARGE CONTROL AGENT, TONER, IMAGE FORMING METHOD, AND IMAGE FORMING APPARATUS CANON KABUSHIKI KAISHA (JP) 2004-07-22 WO disclosed
WO-2004061529-A1 NOVEL POLYHYDROXYALKANOATE HAVING AMIDE, SULFONIC ACID OR SULFONATE ESTER GROUP, CHARGE CONTROL AGENT AND TONER CANON KABUSHIKI KAISHA (JP) 2004-07-22 WO disclosed