SCHEMBL14599985

SCHEMBL14599985

COc1cc(C(C)C)c(OCC#N)cc1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 2/20 0.46
P2RX2 Q9UBL9 2/20 0.46
POLB P06746 1/20 0.45
GAA P10253 1/20 0.45
GFER P55789 1/20 0.45
CYP1A2 P05177 1/20 0.40
ADRA2A P08913 1/20 0.40
CYP2D6 P10635 1/20 0.40
PKM P14618 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
ADRA1D P25100 1/20 0.40
HTR2C P28335 1/20 0.40
ADRA1A P35348 1/20 0.40
HRH1 P35367 1/20 0.40
ADRA1B P35368 1/20 0.40
DRD3 P35462 1/20 0.40
OPRK1 P41145 1/20 0.40
CHRNA4 P43681 1/20 0.40
HIF1A Q16665 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19364184 0.89 P2RX3 (0.42) P2RX3P2RX2POLBGAAGFER
SCHEMBL14566650 0.87 TAAR1 (0.44) POLBGAASMN1; SMN2KDM4ELMNA
SCHEMBL14566485 0.85 ALDH1A1 (0.36) P2RX3P2RX2POLBGAAGFER
SCHEMBL20183061 0.83 ALOX15 (0.40) P2RX3P2RX2POLBGAAGFER
SCHEMBL1493906 0.83 P2RX3 (0.47) P2RX3P2RX2POLBGAAGFER
SCHEMBL2485209 0.83 P2RX3 (0.50) P2RX3P2RX2CYP1A2CYP2D6HTR2C
SCHEMBL1494087 0.83 P2RX3 (0.47) P2RX3P2RX2TAAR1
SCHEMBL12832328 0.80 P2RX3 (0.34) P2RX3P2RX2POLBGAAGFER
Thymoquinol Dimethylether SCHEMBL12613923 0.79 POLB (0.66) P2RX3P2RX2POLBGAAGFER
SCHEMBL13087352 0.79 LMNA (0.43) P2RX3P2RX2POLBGAAGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025898-A1 PROCESS FOR SYNTHESIS OF ARYLOXY DIAMINOPYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 2007-03-08 WO disclosed