SCHEMBL1460131

SCHEMBL1460131

CS(=O)(=O)c1ccc(-c2ccc3c(ccn3-c3c(F)cccc3F)c2)c(C(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 16/20 0.42
KIF11 P52732 1/20 0.42
AR P10275 8/20 0.41
PGR P06401 6/20 0.41
PTGS2 P35354 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1460085 0.73 KIF11 (0.42) NR3C1KIF11ARPGRPTGS2
SCHEMBL28160376 0.70 PTGS2 (0.54) KIF11PTGS2
SCHEMBL585873 0.65 KIF11 (0.60) KIF11ARPTGS2
SCHEMBL28111372 0.64 PTGS2 (0.58) PTGS2
SCHEMBL18751892 0.63 PTGS2 (0.42) NR3C1ARPGRPTGS2
SCHEMBL1460151 0.63 CYP11B1 (0.36) NR3C1PGR
SCHEMBL4011934 0.63 NR1H2 (0.83)
SCHEMBL17394027 0.63 GLA (0.56) KIF11PTGS2
SCHEMBL1460084 0.63 NR3C1 (0.42) NR3C1KIF11ARPGR
SCHEMBL4013753 0.62 NR1H2 (0.80)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011036130-A1 INDOLE DERIVATIVES AS CRAC MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2011-03-31 WO disclosed