SCHEMBL1460410

SCHEMBL1460410

CC(=O)Oc1nn(-c2ccccc2Cl)c(O)c1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.44
RIPK1 Q13546 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
POLB P06746 2/20 0.38
HPGD P15428 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
PDE4A P27815 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
MAPK14 Q16539 2/20 0.36
MAPK11 Q15759 1/20 0.36
WNT3A P56704 1/20 0.36
ALDH1A1 P00352 2/20 0.36
OPRM1 P35372 1/20 0.36
NOTUM Q6P988 1/20 0.35
RARG P13631 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1460386 0.83 PDE4B (0.44) PDE4BRIPK1NPC1RAB9ASMN1; SMN2
SCHEMBL27967501 0.83 MAPK14 (0.43) NPC1RAB9ASMN1; SMN2NPSR1MAPK14
SCHEMBL1722408 0.82 MARS1 (0.37) RIPK1
SCHEMBL1459190 0.81 PDE4B (0.43) PDE4BRIPK1NPC1RAB9ASMN1; SMN2
SCHEMBL2853643 0.75 PDE4B (0.43) PDE4BRIPK1NPC1RAB9ASMN1; SMN2
SCHEMBL27629217 0.69 FABP3 (0.51) ALDH1A1MAPT
SCHEMBL11562429 0.68 SMN1; SMN2 (0.47) PDE4BNPC1RAB9ASMN1; SMN2HPGD
SCHEMBL10698208 0.66 PDE4B (0.42) PDE4BRIPK1NPC1RAB9ASMN1; SMN2
SCHEMBL702658 0.64 CNR1 (0.48)
SCHEMBL4917405 0.64 KDM4E (0.50) PDE4BRIPK1NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349261-A2 PYRAZOLO PYRIDINE DERIVATIVES AS NADPH OXIDASE INHIBITORS GenKyoTex SA (CH) 2011-08-03 EP disclosed
EP-2344492-A1 PYRAZOLO PYRIDINE DERIVATIVES AS NADPH OXIDASE INHIBITORS GenKyoTex SA (CH) 2011-07-20 EP disclosed
EP-2305679-A1 Pyrazoline dione derivatives as nadph oxidase inhibitors GenKyoTex SA (CH) 2011-04-06 EP disclosed
WO-2011036651-A1 PYRAZOLINE DIONE DERIVATIVES AS NADPH OXIDASE INHIBITORS GENKYOTEX SA (CH) 2011-03-31 WO disclosed