SCHEMBL14604384

SCHEMBL14604384

CN(C)C(=O)c1[nH]c2c(-c3ccccc3)c(Cl)ccc2c(=O)c1CN

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAP2 P11137 4/20 0.41
DPP4 P27487 3/20 0.38
MCL1 Q07820 2/20 0.36
ALDH1A1 P00352 2/20 0.35
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
RPA1 P27694 1/20 0.35
PDE10A Q9Y233 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPK8 P45983 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14604052 0.86 MAP2 (0.40) MAP2ALDH1A1LMNASMN1; SMN2KDM4E
SCHEMBL14604429 0.85 PTGS2 (0.45) MAP2MCL1ALDH1A1SMN1; SMN2RPA1
Hydrochloric Acid SCHEMBL14604154 0.85 MAP2 (0.40) MAP2ALDH1A1LMNASMN1; SMN2KDM4E
SCHEMBL14604430 0.83 MAP2 (0.35) MAP2MCL1ALDH1A1LMNASMN1; SMN2
SCHEMBL14604023 0.80 MAPK8 (0.53) SMN1; SMN2MAPK8
SCHEMBL14603988 0.75 MCL1 (0.49) MAP2MCL1ALDH1A1SMN1; SMN2RPA1
SCHEMBL14604161 0.75 MAPK8 (0.39) MAP2ALDH1A1LMNASMN1; SMN2KDM4E
SCHEMBL14604245 0.73 MAPK8 (0.60) ALDH1A1MAPK8
SCHEMBL14604334 0.72 GRIN1 (0.57) MAP2MCL1LMNASMN1; SMN2MAPK8
SCHEMBL12984854 0.71 LMNA (0.44) MAP2MCL1ALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2731932-A1 AMINOMETHYL QUINOLONE COMPOUNDS F.HOFFMANN-LA ROCHE AG (CH) 2014-05-21 EP disclosed
WO-2013007676-A1 AMINOMETHYL QUINOLONE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2013-01-17 WO disclosed