SCHEMBL14615599

SCHEMBL14615599

C=C(NCCc1ccc2ccccc2c1)C(C)(C)N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.46
MAPT P10636 2/20 0.41
CASR P41180 2/20 0.41
RXFP1 Q9HBX9 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2A6 P11509 1/20 0.41
SIGMAR1 Q99720 2/20 0.41
MC4R P32245 2/20 0.41
MC5R P33032 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
HTT P42858 1/20 0.41
IDO1 P14902 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
OPRM1 P35372 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14615486 0.83 CES2 (0.52) CES2MAPTRXFP1CYP1A2KDM4E
SCHEMBL761158 0.74 KDM4E (0.61) CES2MAPTRXFP1CYP1A2KDM4E
SCHEMBL6198665 0.74 CES2 (0.54) CES2MAPTRXFP1CYP1A2MC4R
SCHEMBL12251060 0.73 CYP1A2 (0.50) CES2CASRCYP1A2CYP2A6SIGMAR1
SCHEMBL2732841 0.72 CYP1A2 (0.58) CES2MAPTRXFP1CYP1A2KDM4E
SCHEMBL14748080 0.72 FCER2 (0.55) MC4RMC3R
SCHEMBL3240006 0.72 CES2 (0.66) CES2MAPTRXFP1CYP1A2KDM4E
SCHEMBL13652571 0.72 MTNR1A (0.62) CES2MAPTRXFP1KDM4EALDH1A1
SCHEMBL11822095 0.72 CYP1A2 (0.52) CYP1A2CYP2A6SIGMAR1MC4RMC5R
SCHEMBL2255106 0.71 HDAC1 (0.53) CES2CYP1A2CYP2A6SIGMAR1MC4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007014258-A2 GROWTH HORMONE SECRETAGOGUES SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES S.A.S. (FR) 2007-02-01 WO disclosed