SCHEMBL1461945

SCHEMBL1461945

CCN(Cc1ccccc1)C1CCC(C(O)(C(F)(F)F)C(F)(F)F)CC1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.48
NR1H2 P55055 6/20 0.45
NR1H3 Q13133 6/20 0.45
DPP4 P27487 1/20 0.45
DPP8 Q6V1X1 1/20 0.45
DPP9 Q86TI2 1/20 0.45
DPP7 Q9UHL4 1/20 0.45
SLC6A2 P23975 3/20 0.43
SLC6A4 P31645 3/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
RAB9A P51151 1/20 0.40
LTA4H P09960 1/20 0.39
YTHDC1 Q96MU7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1460723 0.90 DRD2 (0.47) GRIN2BNR1H2NR1H3SLC6A2SLC6A4
SCHEMBL5355490 0.85 SLC6A2 (0.44) GRIN2BNR1H2NR1H3DPP4DPP9
SCHEMBL3371525 0.82 GRIN2B (0.63) GRIN2BDPP4DPP8DPP9DPP7
SCHEMBL21222468 0.81 NR1H2 (0.43) GRIN2BNR1H2NR1H3DPP4DPP8
SCHEMBL21222467 0.81 NR1H2 (0.43) GRIN2BNR1H2NR1H3DPP4DPP8
SCHEMBL1461928 0.80 OPRM1 (0.58) SLC6A2SLC6A4
SCHEMBL1460744 0.79 DPP4 (0.48) DPP4DPP9DPP7SLC6A2SLC6A4
SCHEMBL17139869 0.77 YTHDC1 (0.46) GRIN2BNR1H2NR1H3SLC6A2SLC6A4
SCHEMBL15689171 0.77 YTHDC1 (0.46) GRIN2BNR1H2NR1H3SLC6A2SLC6A4
SCHEMBL15715169 0.77 YTHDC1 (0.46) GRIN2BNR1H2NR1H3SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101087754-B Cyclohexane derivatives HOFFMANN LA ROCHE 2012-01-18 CN claimed
JP-4644714-B2 2011-03-02 JP claimed
JP-2008524280-A 2008-07-10 JP claimed
CN-101087754-A Novel cyclohexane derivatives HOFFMANN LA ROCHE (CH) 2007-12-12 CN claimed
EP-1831158-A1 NOVEL CYCLOHEXANE DERIVATIVES F. Hoffmann-Roche AG (CH) 2007-09-12 EP claimed
US-7253282-B2 Hexafluoroisopropanol substituted cyclohexane derivatives HOFFMAN-LA ROCHE INC. (US) 2007-08-07 US claimed
WO-2006066779-A1 NOVEL CYCLOHEXANE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2006-06-29 WO claimed
US-20060135601-A1 Novel hexafluoroisopropanol substituted cyclohexane derivatives HOFFMANN-LA ROCHE INC. 2006-06-22 US claimed
CN-101087754-B Cyclohexane derivatives HOFFMANN LA ROCHE 2012-01-18 CN disclosed
CN-101087754-A Novel cyclohexane derivatives HOFFMANN LA ROCHE (CH) 2007-12-12 CN disclosed
EP-1831158-A1 NOVEL CYCLOHEXANE DERIVATIVES F. Hoffmann-Roche AG (CH) 2007-09-12 EP disclosed
US-7253282-B2 Hexafluoroisopropanol substituted cyclohexane derivatives HOFFMAN-LA ROCHE INC. (US) 2007-08-07 US disclosed
WO-2006066779-A1 NOVEL CYCLOHEXANE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2006-06-29 WO disclosed
US-20060135601-A1 Novel hexafluoroisopropanol substituted cyclohexane derivatives HOFFMANN-LA ROCHE INC. 2006-06-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060135601-A1 Novel hexafluoroisopropanol substituted cyclohexane derivatives NR1H3, NR1H2, NR1I2 GRIN2B 1121/4885NR1H2 2/4885NR1H3 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.