SCHEMBL14629520

SCHEMBL14629520

CC(C)c1cc(Br)c(O)cc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 4/20 0.43
GABRB1 P18505 2/20 0.43
GABRB2 P47870 2/20 0.41
ADRB2 P07550 2/20 0.40
ADRB1 P08588 1/20 0.40
ADRB3 P13945 1/20 0.40
ADRA1A P35348 3/20 0.38
ADRA2A P08913 2/20 0.38
ADRA2B P18089 2/20 0.38
ADRA2C P18825 2/20 0.38
CYP3A4 P08684 1/20 0.38
HSD17B10 Q99714 1/20 0.38
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
APEX1 P27695 1/20 0.37
RAD52 P43351 1/20 0.37
RECQL P46063 1/20 0.37
BLM P54132 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
KDM4C Q9H3R0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12868984 0.83 GABRA1 (0.43) GABRA1GABRB1GABRB2ADRB2ADRB1
SCHEMBL15631290 0.82 ADRA1A (0.54) GABRA1GABRB1GABRB2ADRB2ADRB1
SCHEMBL5002736 0.80 GABRA1 (0.48) GABRA1GABRB1GABRB2ADRA1ACA1
SCHEMBL5377474 0.80 GABRA1 (0.45) GABRA1GABRB1GABRB2ADRB2ADRB1
SCHEMBL20780493 0.80 LMNA (0.47) GABRA1GABRB1GABRB2ADRB2ADRB1
SCHEMBL24869449 0.80 GABRA1 (0.38) GABRA1GABRB1GABRB2ADRB2CA1
SCHEMBL13484 0.80 GABRA1 (0.38) GABRA1GABRB1GABRB2ADRB2RECQL
SCHEMBL5385858 0.80 GABRA1 (0.48) GABRA1GABRB1GABRB2ADRA1ACYP3A4
SCHEMBL15706603 0.77 LMNA (0.38) GABRA1GABRB1EIF4A3LMNA
SCHEMBL12172238 0.77 LMNA (0.44) GABRA1GABRB2ADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114615981-B KRAS G12D inhibitors 米拉蒂治疗股份有限公司 2024-04-12 CN disclosed
CN-114615981-A KRAS G12D inhibitors 米拉蒂治疗股份有限公司 2022-06-10 CN disclosed
WO-2007005572-A1 PROCESS FOR SYNTHESIZING A CETP INHIBITOR MERCK & CO., INC. (US) 2007-01-11 WO disclosed