SCHEMBL14632005

SCHEMBL14632005

Cc1nc(OC(=O)O)c(-c2ccc(Cl)cc2)s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.48
PTGS1 P23219 2/20 0.46
PTGS2 P35354 2/20 0.46
SMN1; SMN2 Q16637 3/20 0.44
KDM4E B2RXH2 2/20 0.44
RAB9A P51151 2/20 0.44
POLB P06746 2/20 0.44
NPC1 O15118 1/20 0.44
ALDH1A1 P00352 2/20 0.44
PKM P14618 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
ALOX5 P09917 3/20 0.43
MAPT P10636 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
TRPM8 Q7Z2W7 1/20 0.39
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
GAA P10253 1/20 0.38
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27837187 0.88 ALOX5 (0.54) PTGDR2PTGS1PTGS2SMN1; SMN2KDM4E
SCHEMBL14631970 0.88 ALOX5 (0.46) PTGS1PTGS2SMN1; SMN2KDM4ERAB9A
SCHEMBL14631965 0.86 ALOX5 (0.57) PTGS1PTGS2SMN1; SMN2KDM4ERAB9A
SCHEMBL14632061 0.82 KDM4E (0.43) KDM4ENPC1ALDH1A1ALOX5MAPT
SCHEMBL14632042 0.81 ALPL (0.40) SMN1; SMN2ALDH1A1L3MBTL1ALOX5MAPT
SCHEMBL269233 0.77 SMN1; SMN2 (0.51) PTGDR2PTGS1PTGS2SMN1; SMN2KDM4E
SCHEMBL27824201 0.76 ALOX5 (0.56) SMN1; SMN2KDM4ERAB9ANPC1ALOX5
SCHEMBL28790280 0.76 ALOX5 (0.73) PTGS1PTGS2SMN1; SMN2KDM4EALDH1A1
SCHEMBL14632067 0.75 TRPM8 (0.44) SMN1; SMN2KDM4EALOX5TRPM8HCRTR1
SCHEMBL14631942 0.75 ALOX5 (0.44) SMN1; SMN2KDM4ERAB9APOLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188282-B1 1,2-DIAMIDO-ETHYLENE DERIVATIVES AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2013-01-23 EP claimed