SCHEMBL1463333

SCHEMBL1463333

Cn1c(-c2ccccc2)nc2ccccc2c1=O

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.65
KDM4E B2RXH2 2/20 0.62
SMN1; SMN2 Q16637 4/20 0.59
ALDH1A1 P00352 3/20 0.59
CASR P41180 1/20 0.59
RAB9A P51151 2/20 0.58
LMNA P02545 1/20 0.58
RECQL P46063 1/20 0.58
ADRA1A P35348 4/20 0.57
KCNH2 Q12809 4/20 0.57
HRH3 Q9Y5N1 4/20 0.57
MAPT P10636 2/20 0.57
POLB P06746 1/20 0.56
MEN1 O00255 2/20 0.55
HSP90AA1 P07900 1/20 0.55
NPC1 O15118 1/20 0.54
TSHR P16473 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29764078 1.00 KMT2A (0.65) KMT2AKDM4ESMN1; SMN2ALDH1A1CASR
SCHEMBL30311730 0.92 TSHR (0.65) KMT2AKDM4ESMN1; SMN2ALDH1A1RAB9A
SCHEMBL8503249 0.92 TSHR (0.65) KMT2AKDM4ESMN1; SMN2ALDH1A1RAB9A
SCHEMBL14161046 0.89 ADRA1A (0.55) KMT2AKDM4ESMN1; SMN2ALDH1A1ADRA1A
SCHEMBL27926165 0.89 ALDH1A1 (0.60) KMT2AKDM4ESMN1; SMN2ALDH1A1RAB9A
SCHEMBL28639674 0.87 KMT2A (0.57) KMT2AKDM4ESMN1; SMN2ALDH1A1RAB9A
SCHEMBL31276974 0.86 CYP1A2 (0.73) KMT2AKDM4EALDH1A1RAB9ALMNA
SCHEMBL12744507 0.85 KMT2A (0.52) KMT2AKDM4ESMN1; SMN2ALDH1A1LMNA
SCHEMBL31277216 0.84 ADRA1A (0.54) KMT2AKDM4ESMN1; SMN2ALDH1A1ADRA1A
SCHEMBL31277167 0.83 PARG (0.56) KMT2AKDM4ESMN1; SMN2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115650924-B Green synthesis method of quinazolinone 山东华泰新材料技术研发有限公司 2024-08-20 CN disclosed
CN-117964560-A Method for constructing quinazolinone derivative through oxidization 淮阴工学院 2024-05-03 CN disclosed
CN-113563272-B Preparation method of 2-phenylquinazolinone compound 三峡大学 2023-03-10 CN disclosed
CN-115650924-A Green synthesis method of quinazolinone 上海橡实化学有限公司 2023-01-31 CN disclosed
CN-113185468-B Method for synthesizing quinazolinone through photocatalysis 上海橡实化学有限公司 2022-08-26 CN disclosed
CN-113563272-A Preparation method of 2-phenylquinazolinone compound 三峡大学 2021-10-29 CN disclosed
CN-113461617-A Method for preparing N-heterocycle through visible light mediated dehydrogenation 石河子大学 2021-10-01 CN disclosed
CN-113185468-A Method for synthesizing quinazolinone through photocatalysis 上海橡实化学有限公司 2021-07-30 CN disclosed
CN-104557738-A Green synthesis method of 4(3H)-quinazolinone UNIV HUNAN 2015-04-29 CN disclosed
CN-103408502-A Synthetic method of quinazolinone compounds UNIV HUNAN 2013-11-27 CN disclosed
US-20130059869-A1 METHODS AND COMPOSITIONS FOR TREATING DISORDERS HYDRA BIOSCIENCES, INC. 2013-03-07 US disclosed
US-20110071148-A1 COMPOUNDS AS THE ESTROGEN RELATED RECEPTORS MODULATORS AND THE USES THEREOF GUANGZHOU INSTITUTE OF BIOMEDICINE AND HEALTH, CHINESE ACADEMY OF SCIENCES (CN) 2011-03-24 US disclosed
EP-2266962-A1 THE COMPOUNDS AS THE ESTROGEN RELATED RECEPTORS MODULATORS AND THE USES THEREOF Guangzhou Institute Of Biomedicine And Health, Chinese Academy Of Sciences (CN) 2010-12-29 EP disclosed
CN-101531638-A Compounds useful as estrogen-related receptor modulators and uses thereof CHINESE ACADEMY OF SCIENCES GU 2009-09-16 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110071148-A1 COMPOUNDS AS THE ESTROGEN RELATED RECEPTORS MODULATORS AND THE USES THEREOF ESRRA, ESRRB, ESRRG KMT2A 1845/4885KDM4E 1222/4885SMN1; SMN2 4538/4885
US-20130059869-A1 METHODS AND COMPOSITIONS FOR TREATING DISORDERS TRPA1, TRPV1, TRPV3 KMT2A 4200/4885KDM4E 4704/4885SMN1; SMN2 129/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.