SCHEMBL1463944

SCHEMBL1463944

Cc1nccnc1C(N)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.42
MKNK2 Q9HBH9 1/20 0.42
SIRT3 Q9NTG7 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
ADORA3 P0DMS8 2/20 0.40
TSHR P16473 1/20 0.40
MC4R P32245 1/20 0.40
ADRA1A P35348 1/20 0.40
MC3R P41968 1/20 0.40
LMNA P02545 2/20 0.39
KDM4E B2RXH2 2/20 0.39
ADORA2A P29274 2/20 0.39
ADORA1 P30542 2/20 0.39
PKM P14618 1/20 0.39
ADORA2B P29275 1/20 0.39
KAT2B Q92831 1/20 0.39
ALDH1A1 P00352 2/20 0.37
P2RX7 Q99572 1/20 0.37
NNMT P40261 3/20 0.36
PRKCI P41743 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2310300 1.00 MKNK1 (0.42) MKNK1MKNK2SIRT3TDP1ADORA3
SCHEMBL2492969 0.82 TSHR (0.48) SIRT3ADORA3TSHRMC4RADRA1A
SCHEMBL5518273 0.80 KDM4E (0.36) MKNK1MKNK2TSHRKDM4EPKM
SCHEMBL29364216 0.78 SMN1; SMN2 (0.39) MKNK1MKNK2TSHRKDM4EPKM
SCHEMBL287450 0.78 KDM4E (0.47) TSHRKDM4EPKMALDH1A1MAPT
SCHEMBL23864829 0.78 KDM4E (0.35) MKNK1MKNK2TSHRKDM4EPKM
SCHEMBL29526925 0.78 KDM4E (0.47) TSHRKDM4EPKMALDH1A1MAPT
SCHEMBL13544700 0.78 ADORA3 (0.41) SIRT3TDP1ADORA3TSHRMC4R
SCHEMBL335305 0.78 SMN1; SMN2 (0.39) MKNK1MKNK2TSHRKDM4EPKM
SCHEMBL23032651 0.76 KDM4E (0.34) MKNK1MKNK2TSHRKDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026107422-A1 6-(PYRIDIN-4-YL)-1H-BENZO[D]IMIDAZOLE DERIVATIVES AS CAMK2 INHIBITORS FOR THE TREATMENT OF HEART FAILURE BRISTOL-MYERS SQUIBB COMPANY (US) 2026-05-21 WO disclosed
US-12459927-B2 Plasma kallikrein inhibitors MERCK SHARP & DOHME LLC (US) 2025-11-04 US disclosed
US-20240228501-A1 IMIDAZOLE-CONTAINING CONDENSED RING DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF IN MEDICINE CHANGCHUN GENESCIENCE PHARMACEUTICAL CO., LTD. (CN) 2024-07-11 US disclosed
EP-4293023-A1 IMIDAZOLE-CONTAINING CONDENSED RING DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF IN MEDICINE Changchun Genescience Pharmaceutical Co., Ltd. (CN) 2023-12-20 EP disclosed
WO-2022222963-A1 IMIDAZOLE-CONTAINING CONDENSED RING DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF IN MEDICINE 长春金赛药业有限责任公司 2022-10-27 WO disclosed
US-20110071150-A1 INDOLE DERIVATIVES AS CRAC MODULATORS ALAM MUZAFFAR 2011-03-24 US disclosed
US-7728025-B2 2-heteroaryl-substituted benzimidazole derivative BANYU PHARMACEUTICAL CO., LTD. (JP) 2010-06-01 US disclosed
US-20080070928-A1 Novel 2-Heteroaryl-Substituted Benzimidazole Derivative MSD K.K. (JP) 2008-03-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110071150-A1 INDOLE DERIVATIVES AS CRAC MODULATORS ORAI1, RYR2, CACNA1E MKNK1 2518/4885MKNK2 2157/4885SIRT3 1243/4885
US-20080070928-A1 Novel 2-Heteroaryl-Substituted Benzimidazole Derivative GCK, GCKR, HK1 MKNK1 1678/4885MKNK2 1205/4885SIRT3 88/4885
US-20240228501-A1 IMIDAZOLE-CONTAINING CONDENSED RING DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF IN MEDICINE KISS1R, CYP3A43, SLC6A11 MKNK1 2023/4885MKNK2 2767/4885SIRT3 358/4885
US-12459927-B2 Plasma kallikrein inhibitors KLKB1, SERPINE1, KLK5 MKNK1 373/4885MKNK2 559/4885SIRT3 1050/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.