SCHEMBL1464569

SCHEMBL1464569

CCCCc1ccc(C(=O)Nc2ccccc2C(=O)C(O)c2ccccc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 15/20 0.66
PLK3 Q9H4B4 7/20 0.66
TRPV1 Q8NER1 3/20 0.58
ABCG2 Q9UNQ0 1/20 0.49
SLC16A3 O15427 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1464667 0.84 PLK1 (0.90) PLK1PLK3TRPV1SLC16A3
SCHEMBL6838813 0.81 CES2 (0.59) PLK1TRPV1
SCHEMBL28808948 0.81 PLK1 (0.97) PLK1PLK3
SCHEMBL15170179 0.80 BACE1 (0.59)
SCHEMBL6837052 0.78 CES2 (0.57) TRPV1
SCHEMBL23657651 0.76 TRPV1 (0.68) PLK1PLK3TRPV1
SCHEMBL6836519 0.76 RARB (0.56)
SCHEMBL6836850 0.76 RARB (0.56)
SCHEMBL6832878 0.76 RARB (0.56)
SCHEMBL6838814 0.76 CES2 (0.59) PLK1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110071197-A1 BIS-ARYL COMPOUNDS FOR USE AS MEDICAMENTS BIOLIPOX AB (LV) 2011-03-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110071197-A1 BIS-ARYL COMPOUNDS FOR USE AS MEDICAMENTS LTC4S, LTB4R2, LTB4R PLK1 3734/4885PLK3 1566/4885TRPV1 377/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.