SCHEMBL14647203

SCHEMBL14647203

Cc1ccc2c(c1)OCCN2C1CCOCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM5 P08912 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
KCNH2 Q12809 1/20 0.38
PIK3CB P42338 2/20 0.37
PIK3CG P48736 2/20 0.37
PIK3CD O00329 1/20 0.37
GRIA2 P42262 1/20 0.36
HTR1A P08908 1/20 0.35
HTR1D P28221 1/20 0.35
HTR1F P30939 1/20 0.35
ALDH1A1 P00352 1/20 0.35
PRKDC P78527 1/20 0.35
AVPR1A P37288 2/20 0.35
AVPR1B P47901 1/20 0.35
PIK3CA P42336 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14647199 0.86 MEN1 (0.37) PIK3CBPIK3CGPIK3CDGRIA2HTR1A
SCHEMBL24629797 0.82 GAA (0.45) HTR1AHTR1DHTR1FALDH1A1AVPR1A
SCHEMBL566036 0.82 LMNA (0.46) PIK3CBPIK3CGPIK3CDHTR1AHTR1D
SCHEMBL29769101 0.82 GAA (0.45) HTR1AHTR1DHTR1FALDH1A1AVPR1A
SCHEMBL16440168 0.79 AAK1 (0.43)
SCHEMBL24629796 0.79 HTR1A (0.40) HTR1AHTR1DHTR1FALDH1A1MEN1
SCHEMBL2018716 0.78 HTR2C (0.47)
SCHEMBL692930 0.78 HTR2C (0.47)
SCHEMBL29769185 0.77 ALDH1A1 (0.48) ALDH1A1
SCHEMBL29769100 0.77 MAPT (0.55) HTR1AHTR1DHTR1FALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022150574-A1 INHIBITORS OF MYCOBACTERIUM TUBERCULOSIS LIPOAMIDE DEHYDROGENASE CORNELL UNIVERSITY (US) 2022-07-14 WO disclosed
EP-2373649-B1 INDOLE AND BENZOXAZINE DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS JANSSEN PHARMACEUTICALS INC (US) 2013-01-23 EP disclosed